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A review on synthesis, mechanism of action, and structure-activity relationships of 1, 2, 3-triazole-based α-glucosidase inhibitors as promising anti-diabetic agents
Abstract α-Glucosidase is a key enzyme in hydrolysis of carbohydrates to glucose and
located in the small intestine brush border. Inhibition of this enzyme delay the release of …
located in the small intestine brush border. Inhibition of this enzyme delay the release of …
Recent advances of α-glucosidase inhibitors: a comprehensive review
Background: Diabetes mellitus (DM) is a critical health issue prevailing in nearly half a
billion people worldwide. It is one of the most threatening metabolic diseases. Type 2 DM is …
billion people worldwide. It is one of the most threatening metabolic diseases. Type 2 DM is …
Design and synthesis of novel quinazolinone-1, 2, 3-triazole hybrids as new anti-diabetic agents: In vitro α-glucosidase inhibition, kinetic, and docking study
A novel series of quinazolinone-1, 2, 3-triazole hybrids 10a-p were designed, synthesized,
and evaluated for their in vitro α-glucosidase inhibitory activity leading to efficient anti …
and evaluated for their in vitro α-glucosidase inhibitory activity leading to efficient anti …
Synthesis, anticancer activity and molecular docking of new quinolines, quinazolines and 1, 2, 4-triazoles with pyrido [2, 3-d] pyrimidines
Recently, heterocyclic compounds such as pyrido [2, 3-d] pyrimidinones, 1, 2, 4-
triazolopyrimidines, pyrimidoquinazolines, and quinoline derivatives have gained attention …
triazolopyrimidines, pyrimidoquinazolines, and quinoline derivatives have gained attention …
Discovery of triazole tethered thymol/carvacrol-coumarin hybrids as new class of α-glucosidase inhibitors with potent in vivo antihyperglycemic activities
Kee** in view the inhibitory potential of monoterpenes thymol and carvacrol as well as
coumarin nucleus against α-glucosidase, novel series of thymol/carvacrol-coumarin hybrids …
coumarin nucleus against α-glucosidase, novel series of thymol/carvacrol-coumarin hybrids …
Evaluation of novel 2-(quinoline-2-ylthio) acetamide derivatives linked to diphenyl-imidazole as α-glucosidase inhibitors: Insights from in silico, in vitro, and in vivo …
The inhibition of the α-glucosidase enzyme is crucial for targeting type 2 diabetes mellitus
(DM). This study introduces a series of synthetic analogs based on thiomethylacetamide …
(DM). This study introduces a series of synthetic analogs based on thiomethylacetamide …
Biscoumarin-1, 2, 3-triazole hybrids as novel anti-diabetic agents: Design, synthesis, in vitro α-glucosidase inhibition, kinetic, and docking studies
A novel series of biscoumarin-1, 2, 3-triazole hybrids 6a-n was prepared and evaluated for α-
glucosidase inhibitory potential. All fourteen derivatives exhibited excellent α-glucosidase …
glucosidase inhibitory potential. All fourteen derivatives exhibited excellent α-glucosidase …
Arylureidoaurones: Synthesis, in vitro α-glucosidase, and α-amylase inhibition activity
M Kazempour-Dizaji, S Mojtabavi, A Sadri… - Bioorganic …, 2023 - Elsevier
Because of the colossal global burden of diabetes, there is an urgent need for more effective
and safer drugs. We designed and synthesized a new series of aurone derivatives …
and safer drugs. We designed and synthesized a new series of aurone derivatives …
Synthesis, characterization, molecular docking, and biological activities of coumarin–1, 2, 3‐triazole‐acetamide hybrid derivatives
Coumarins and their derivatives are receiving increasing attention due to numerous
biochemical and pharmacological applications. In this study, a series of novel coumarin–1 …
biochemical and pharmacological applications. In this study, a series of novel coumarin–1 …
Synthesis and biological evaluation of new benzimidazole-1, 2, 3-triazole hybrids as potential α-glucosidase inhibitors
N Asemanipoor, M Mohammadi-Khanaposhtani… - Bioorganic …, 2020 - Elsevier
In this study, a series of benzimidazole-1, 2, 3-triazole hybrids 8a-n as new α-glucosidase
inhibitors were designed and synthesized. In vitro α-glucosidase inhibition activity results …
inhibitors were designed and synthesized. In vitro α-glucosidase inhibition activity results …