[HTML][HTML] Recent development on COX-2 inhibitors as promising anti-inflammatory agents: The past 10 years

Z Ju, M Li, J Xu, DC Howell, Z Li, FE Chen - Acta Pharmaceutica Sinica B, 2022‏ - Elsevier
Cyclooxygenases play a vital role in inflammation and are responsible for the production of
prostaglandins. Two cyclooxygenases are described, the constitutive cyclooxygenase-1 and …

[HTML][HTML] An overview of the biological evaluation of selected nitrogen-containing heterocycle medicinal chemistry compounds

O Ebenezer, MA Jordaan, G Carena, T Bono… - International Journal of …, 2022‏ - mdpi.com
Heterocyclic compounds are a class of compounds of natural origin with favorable
properties and hence have major pharmaceutical significance. They have an exceptional …

Design, characterization and in vivo performance of solid lipid nanoparticles (SLNs)-loaded mucoadhesive buccal tablets for efficient delivery of Lornoxicam in …

MB Zewail, GF Asaad, SM Swellam… - International Journal of …, 2022‏ - Elsevier
Lornoxicam (LRX) is a potent nonsteroidal anti-inflammatory drug (NSAID) used extensively
to manage pain and inflammatory conditions. However, the drug possesses poor aqueous …

Design, synthesis, and antiproliferative properties of new 1, 2, 3-triazole-carboximidamide derivatives as dual EGFR/VEGFR-2 inhibitors

MA Mahmoud, AF Mohammed, OIA Salem… - Journal of Molecular …, 2023‏ - Elsevier
A new series of substituted aryl carboximidamide VIa-o was designed and synthesised. IR, 1
H NMR, 13 C NMR as well as elemental microanalysis were used to confirm the structures of …

A comprehensive review of recent advances in the biological activities of 1, 2, 4‐oxadiazoles

OM Hendawy - Archiv der Pharmazie, 2022‏ - Wiley Online Library
Nitrogen heterocycles play an essential role in medication development. The 1, 2, 4‐
oxadiazole heterocycle has been extensively studied, yielding a large variety of molecules …

Exploring thiazole-based Schiff base analogs as potent α-glucosidase and α-amylase inhibitor: their synthesis and in-silico study

M Taha, S Hayat, F Rahim, N Uddin, A Wadood… - Journal of Molecular …, 2023‏ - Elsevier
In search of potent antidiabetic agents here in this study a new series of thiazole-based
Schiff base analogs (1–20) have been synthesized, characterized by 1 HNMR, 13 CNMR …

[HTML][HTML] Synthesis and biological evaluation of indole-2-carboxamides with potent apoptotic antiproliferative activity as egfr/cdk2 dual inhibitors

LH Al-Wahaibi, YA Mostafa, MH Abdelrahman… - Pharmaceuticals, 2022‏ - mdpi.com
The apoptotic antiproliferative actions of our previously reported CB1 allosteric modulators 5-
chlorobenzofuran-2-carboxamide derivatives VIIa–j prompted us to develop and synthesise …

[HTML][HTML] A review on progress of thiazole derivatives as potential anti-inflammatory agents

KH Narasimhamurthy, TR Swaroop… - European Journal of …, 2024‏ - Elsevier
Inflammation is a body response against infection that activates other biological components
that include various cytokines, chemokines and other biological compounds that trigger …

Design and synthesis of new dihydropyrimidine/sulphonamide hybrids as promising anti-inflammatory agents via dual mPGES-1/5-LOX inhibition

LH Al-Wahaibi, AM Elshamsy, TFS Ali… - Frontiers in …, 2024‏ - frontiersin.org
A novel series of dihydropyrimidine/sulphonamide hybrids 3a–j with anti-inflammatory
properties have been developed and tested as dual mPGES-1/5-LOX inhibitors. In vitro …

Design, Synthesis, and Anti-Proliferative Action of Purine/Pteridine-Based Derivatives as Dual Inhibitors of EGFR and BRAFV600E

SA El-Kalyoubi, HAM Gomaa, EMN Abdelhafez… - Pharmaceuticals, 2023‏ - mdpi.com
The investigation of novel EGFR and BRAFV600E dual inhibitors is intended to serve as
targeted cancer treatment. Two sets of purine/pteridine-based derivatives were designed …