End-point binding free energy calculation with MM/PBSA and MM/GBSA: strategies and applications in drug design

E Wang, H Sun, J Wang, Z Wang, H Liu… - Chemical …, 2019 - ACS Publications
Molecular mechanics Poisson–Boltzmann surface area (MM/PBSA) and molecular
mechanics generalized Born surface area (MM/GBSA) are arguably very popular methods …

How water's properties are encoded in its molecular structure and energies

E Brini, CJ Fennell, M Fernandez-Serra… - Chemical …, 2017 - ACS Publications
How are water's material properties encoded within the structure of the water molecule? This
is pertinent to understanding Earth's living systems, its materials, its geochemistry and …

[HTML][HTML] A guide to in silico drug design

Y Chang, BA Hawkins, JJ Du, PW Groundwater… - Pharmaceutics, 2023 - mdpi.com
The drug discovery process is a rocky path that is full of challenges, with the result that very
few candidates progress from hit compound to a commercially available product, often due …

Assessing the performance of the MM/PBSA and MM/GBSA methods. 1. The accuracy of binding free energy calculations based on molecular dynamics simulations

T Hou, J Wang, Y Li, W Wang - Journal of chemical information …, 2011 - ACS Publications
The Molecular Mechanics/Poisson− Boltzmann Surface Area (MM/PBSA) and the Molecular
Mechanics/Generalized Born Surface Area (MM/GBSA) methods calculate binding free …

SIRT4 is a lysine deacylase that controls leucine metabolism and insulin secretion

KA Anderson, FK Huynh, K Fisher-Wellman, JD Stuart… - Cell metabolism, 2017 - cell.com
Sirtuins are NAD+-dependent protein deacylases that regulate several aspects of
metabolism and aging. In contrast to the other mammalian sirtuins, the primary enzymatic …

The VSGB 2.0 model: a next generation energy model for high resolution protein structure modeling

J Li, R Abel, K Zhu, Y Cao, S Zhao… - Proteins: Structure …, 2011 - Wiley Online Library
A novel energy model (VSGB 2.0) for high resolution protein structure modeling is
described, which features an optimized implicit solvent model as well as physics‐based …

Identification of post-digestion angiotensin-I converting enzyme (ACE) inhibitory peptides from soybean protein Isolate: Their production conditions and in silico …

Z Xu, C Wu, D Sun-Waterhouse, T Zhao… - Food Chemistry, 2021 - Elsevier
This study attempts to investigate natural angiotensin-I converting enzyme (ACE) inhibitors.
Soybean protein isolated (SPI) hydrolysate (SPIH) was prepared by Alcalase from …

The Amber biomolecular simulation programs

DA Case, TE Cheatham III, T Darden… - Journal of …, 2005 - Wiley Online Library
We describe the development, current features, and some directions for future development
of the Amber package of computer programs. This package evolved from a program that was …

CHARMM: the biomolecular simulation program

BR Brooks, CL Brooks III… - Journal of …, 2009 - Wiley Online Library
Abstract CHARMM (Chemistry at HARvard Molecular Mechanics) is a highly versatile and
widely used molecular simulation program. It has been developed over the last three …

[PDF][PDF] Amber 10

DA Case, TA Darden, TE Cheatham, CL Simmerling… - 2008 - infoscience.epfl.ch
Amber is the collective name for a suite of programs that allow users to carry out molecular
dynamics simulations, particularly on biomolecules. None of the individual programs carries …