Turnitin
降AI改写
早检测系统
早降重系统
Turnitin-UK版
万方检测-期刊版
维普编辑部版
Grammarly检测
Paperpass检测
checkpass检测
PaperYY检测
Recent advances of imidazole-containing derivatives as anti-tubercular agents
YL Fan, XH **, ZP Huang, HF Yu, ZG Zeng… - European journal of …, 2018 - Elsevier
Tuberculosis still remains one of the most common, communicable, and leading deadliest
diseases known to mankind throughout the world. Drug-resistance in Mycobacterium …
diseases known to mankind throughout the world. Drug-resistance in Mycobacterium …
Prodrug design to improve pharmacokinetic and drug delivery properties: challenges to the discovery scientists
The prodrug design is a versatile, powerful method that can be applied to a wide range of
parent drug molecules, administration routes, and formulations. Clinically, the majority of …
parent drug molecules, administration routes, and formulations. Clinically, the majority of …
Nitro-group-containing drugs
The nitro group is considered to be a versatile and unique functional group in medicinal
chemistry. Despite a long history of use in therapeutics, the nitro group has toxicity issues …
chemistry. Despite a long history of use in therapeutics, the nitro group has toxicity issues …
Photoredox cross-coupling: Ir/Ni dual catalysis for the synthesis of benzylic ethers
Single-electron transmetalation has emerged as an enabling paradigm for the cross-
coupling of Csp3 hybridized organotrifluoroborates. Cross-coupling of α …
coupling of Csp3 hybridized organotrifluoroborates. Cross-coupling of α …
Antituberculosis drug research: a critical overview
The increasing drug resistance of M ycobacterium tuberculosis to the currently used drugs
and HIV coinfection has caused alarm in the international scientific community …
and HIV coinfection has caused alarm in the international scientific community …
An efficient one-pot synthesis of heterocycle-fused 1, 2, 3-triazole derivatives as anti-cancer agents
SJ Yan, YJ Liu, YL Chen, L Liu, J Lin - Bioorganic & Medicinal Chemistry …, 2010 - Elsevier
A series of heterocycle-fused 1, 2, 3-triazoles were easily prepared by the 1, 3-dipolar
cycloaddition of heterocyclic ketene aminals or N, O-acetals with sodium azide and polyhalo …
cycloaddition of heterocyclic ketene aminals or N, O-acetals with sodium azide and polyhalo …
Prodrugs: bridging pharmacodynamic/pharmacokinetic gaps
B Testa - Current opinion in chemical biology, 2009 - Elsevier
In this mini review, prodrugs are discussed with a focus on their pharmaceutical,
pharmacokinetic, and pharmacodynamic objectives, as well as on the resulting therapeutic …
pharmacokinetic, and pharmacodynamic objectives, as well as on the resulting therapeutic …
[HTML][HTML] Nitroaromatic antibiotics as nitrogen oxide sources
Nitroaromatic antibiotics show activity against anaerobic bacteria and parasites, finding use
in the treatment of Heliobacter pylori infections, tuberculosis, trichomoniasis, human African …
in the treatment of Heliobacter pylori infections, tuberculosis, trichomoniasis, human African …
Nitroimidazoles for the treatment of TB: past, present and future
T Mukherjee, H Boshoff - Future medicinal chemistry, 2011 - Taylor & Francis
Tuberculosis remains a leading cause of death resulting from an infectious agent, and the
spread of multi-and extensively drug-resistant strains of Mycobacterium tuberculosis poses a …
spread of multi-and extensively drug-resistant strains of Mycobacterium tuberculosis poses a …
Highly enantioselective, hydrogen-bond-donor catalyzed additions to oxetanes
A precisely designed chiral squaramide derivative is shown to promote the highly
enantioselective addition of trimethylsilyl bromide (TMSBr) to a broad variety of 3-substituted …
enantioselective addition of trimethylsilyl bromide (TMSBr) to a broad variety of 3-substituted …