Structural basis of potential inhibitors targeting SARS-CoV-2 main protease

HM Mengist, T Dilnessa, T ** - Frontiers in Chemistry, 2021 - frontiersin.org
The Coronavirus disease-19 (COVID-19) pandemic is still devastating the world causing
significant social, economic, and political chaos. Corresponding to the absence of globally …

Repurposing drugs for the management of COVID-19

J Cusinato, Y Cau, AM Calvani… - Expert opinion on …, 2021 - Taylor & Francis
Introduction: The coronavirus disease 2019 (COVID-19) caused by SARS-CoV-2 represents
a serious health issue worldwide, with more than 61 million cases and more than 1.4 million …

Methodology-centered review of molecular modeling, simulation, and prediction of SARS-CoV-2

K Gao, R Wang, J Chen, L Cheng, J Frishcosy… - Chemical …, 2022 - ACS Publications
Despite tremendous efforts in the past two years, our understanding of severe acute
respiratory syndrome coronavirus 2 (SARS-CoV-2), virus–host interactions, immune …

[HTML][HTML] An overview of potential inhibitors targeting non-structural proteins 3 (PLpro and Mac1) and 5 (3CLpro/Mpro) of SARS-CoV-2

F Yan, F Gao - Computational and structural biotechnology journal, 2021 - Elsevier
There is an urgent need to develop effective treatments for coronavirus disease 2019
(COVID-19), which is caused by severe acute respiratory syndrome coronavirus 2 (SARS …

Computer aided identification of potential SARS CoV-2 main protease inhibitors from diterpenoids and biflavonoids of Torreya nucifera leaves

R Ghosh, A Chakraborty, A Biswas… - Journal of Biomolecular …, 2022 - Taylor & Francis
SARS CoV-2 is the causative agent of the pandemic disease COVID-19. There is an urgent
need for effective drugs or vaccines which can effectively combat this outbreak. The main …

Docking covalent targets for drug discovery: stimulating the computer-aided drug design community of possible pitfalls and erroneous practices

AQK Oyedele, AT Ogunlana, ID Boyenle… - Molecular Diversity, 2023 - Springer
The continuous approval of covalent drugs in recent years for the treatment of diseases has
led to an increased search for covalent agents by medicinal chemists and computational …

Molecular docking as a potential approach in repurposing drugs against COVID-19: A systematic review and novel pharmacophore models

M Fadlalla, M Ahmed, M Ali, AA Elshiekh… - Current Pharmacology …, 2022 - Springer
Abstract Purpose of Review This article provides a review of the recent literature related to
the FDA-approved drugs that had been repurposed as potential drug candidates against …

Phytochemical rich Himalayan Rhododendron arboreum petals inhibit SARS-CoV-2 infection in vitro

M Lingwan, S Shagun, F Pahwa, A Kumar… - Journal of …, 2023 - Taylor & Francis
Phytochemicals with potential to competitively bind to the host receptors or inhibit SARS-
CoV-2 replication, may prove to be useful as adjunct therapeutics for COVID-19. We profiled …

A survey on computational methods in discovering protein inhibitors of SARS-CoV-2

Q Liu, J Wan, G Wang - Briefings in Bioinformatics, 2022 - academic.oup.com
The outbreak of acute respiratory disease in 2019, namely Coronavirus Disease-2019
(COVID-19), has become an unprecedented healthcare crisis. To mitigate the pandemic …

SARS-CoV-2 entry inhibitors by dual targeting TMPRSS2 and ACE2: An in silico drug repurposing study

K Baby, S Maity, CH Mehta, A Suresh, UY Nayak… - European Journal of …, 2021 - Elsevier
Abstract The coronavirus disease (COVID-19) is spreading between human populations
mainly through nasal droplets. Currently, the vaccines have great hope, but it takes years for …