The role of inflammasomes in human diseases and their potential as therapeutic targets

J Yao, K Sterling, Z Wang, Y Zhang… - Signal Transduction and …, 2024 - nature.com
Inflammasomes are large protein complexes that play a major role in sensing inflammatory
signals and triggering the innate immune response. Each inflammasome complex has three …

[HTML][HTML] Advances in the roles of ATF4 in osteoporosis

Y **ao, X **e, Z Chen, G Yin, W Kong, J Zhou - Biomedicine & …, 2023 - Elsevier
Osteoporosis (OP) is characterized by reduced bone mass, decreased strength, and
enhanced bone fragility fracture risk. Activating transcription factor 4 (ATF4) plays a role in …

Design, Synthesis, and Biological Evaluation of Ferulic Acid-Piperazine Derivatives Targeting Pathological Hallmarks of Alzheimer's Disease

G Singh, S Kumar, SR Panda, P Kumar… - ACS Chemical …, 2024 - ACS Publications
Alzheimer's disease (AD) is the most prevalent cause of dementia and is characterized by
low levels of acetyl and butyrylcholine, increased oxidative stress, inflammation …

Gingerenone A Attenuates Ulcerative Colitis via Targeting IL‐17RA to Inhibit Inflammation and Restore Intestinal Barrier Function

J Liang, W Dai, C Liu, Y Wen, C Chen, Y Xu… - Advanced …, 2024 - Wiley Online Library
Ulcerative colitis (UC) is a complicated and recurrent intestinal disease. Currently available
drugs for UC treatment are scarce, therefore, novel therapeutic drugs for the UC are urgently …

Tabersonine, a natural NLRP3 inhibitor, suppresses inflammasome activation in macrophages and attenuate NLRP3-driven diseases in mice

H Xu, W Li, S Hong, J Shao, J Chen… - Acta Pharmacologica …, 2023 - nature.com
Aberrant activation of NLRP3 inflammasome causes the progression of various inflammation-
related diseases, but the small-molecule inhibitors of NLRP3 are not currently available for …

Target discovery of bioactive natural products with Native-compound-Coupled CNBr-activated Sepharose 4B Beads (NCCB): applications, mechanisms and outlooks

Y Zhang, J Zhang, M Li, Y Qiao, W Wang, L Ma… - Bioorganic & Medicinal …, 2023 - Elsevier
Natural products (NPs) represent a treasure trove for drug discovery and development due
to their chemical structural diversity and a broad spectrum of biological activities. Uncovering …

Mesenchymal stem cells and their extracellular vesicles in bone and joint diseases: targeting the NLRP3 inflammasome

S Xu, Y Zhang, Z Zheng, J Sun, Y Wei, G Ding - Human Cell, 2024 - Springer
The nucleotide-binding oligomerization domain-like-receptor family pyrin domain-containing
3 (NLRP3) inflammasome is a cytosolic multi-subunit protein complex, and recent studies …

A natural sesquiterpene lactone isolinderalactone attenuates lipopolysaccharide-induced inflammatory response and acute lung injury through inhibition of NF-κB …

X Shen, H Chen, H Zhang, L Luo, T Wen, L Liu… - International …, 2023 - Elsevier
Isolinderalactone is the main sesquiterpene lactone isolated from Lindera aggregata, a
traditional Chinese medicine widely used to treat pain and inflammation. Although …

Novel MAGL inhibitors alleviate LPS-induced acute kidney injury by inhibiting NLRP3 inflammatory vesicles, modulating intestinal flora, repairing the intestinal barrier …

H **ang, Y Wang, L Yang, M Liu, C Sun, Y Gu, J Yao - Molecules, 2023 - mdpi.com
Acute kidney injury (AKI) is a complication of a wide range of serious illnesses for which
there is still no better therapeutic agent. We demonstrated that M-18C has a favorable …

Protective effects of sinomenine against dextran sulfate sodium-induced ulcerative colitis in rats via alteration of HO-1/Nrf2 and inflammatory pathway

Z Niu, X Li, X Yang, Z Sun - Inflammopharmacology, 2024 - Springer
Abstract Background Dextran Sulfate Sodium (DSS) induces ulcerative colitis (UC), a type of
inflammatory bowel disease (IBD) that leads to inflammation, swelling, and ulcers in the …