Glial polarization in neurological diseases: Molecular mechanisms and therapeutic opportunities

Y Liu, L Wu, W Peng, X Mao - Ageing Research Reviews, 2024 - Elsevier
Glial cell polarization plays a pivotal role in various neurological disorders. In response to
distinct stimuli, glial cells undergo polarization to either mitigate neurotoxicity or facilitate …

Effects of low-dose acetylsalicylic acid on the inflammatory response to experimental sleep restriction in healthy humans

LC Engert, C Ledderose, C Biniamin, P Birriel… - Brain, Behavior, and …, 2024 - Elsevier
Background Sleep deficiencies, such as manifested in short sleep duration or insomnia
symptoms, are known to increase the risk for multiple disease conditions involving …

Synthesis and anti‐inflammatory activity of novel firocoxib analogues with balanced COX inhibition

J Xu, K Tang, Z Ju - Chemical Biology & Drug Design, 2024 - Wiley Online Library
The adverse effects caused by nonselective and selective cyclooxygenase‐2 (COX‐2)
inhibitors remain a challenge for current anti‐inflammatory medications. A balanced …

A further pocket or conformational plasticity by map** COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet …

R Solidoro, M Miciaccia, C Bonaccorso… - European Journal of …, 2024 - Elsevier
Cyclooxygenase enzymes have distinct roles in cardiovascular, neurological, and
neurodegenerative disease. They are differently expressed in different type of cancers …

Heterocycle-guided synthesis of m-hetarylanilines via three-component benzannulation

AR Galeev, MV Dmitriev, AS Novikov… - Beilstein Journal of …, 2024 - beilstein-journals.org
A one-pot three-component synthesis of substituted meta-hetarylanilines from heterocycle-
substituted 1, 3-diketones has been developed. The electron-withdrawing power of the …