Overcoming endocrine resistance in breast cancer

AB Hanker, DR Sudhan, CL Arteaga - Cancer cell, 2020‏ - cell.com
Estrogen receptor-positive (ER+) breast cancer is the most common breast cancer subtype.
Treatment of ER+ breast cancer comprises interventions that suppress estrogen production …

[HTML][HTML] PI3K/AKT/mTOR-targeted therapy for breast cancer

K Zhu, Y Wu, P He, Y Fan, X Zhong, H Zheng, T Luo - Cells, 2022‏ - mdpi.com
Phosphatidylinositol 3-kinase (PI3K), protein kinase B (PKB/AKT) and mechanistic target of
rapamycin (mTOR)(PAM) pathways play important roles in breast tumorigenesis and confer …

Proteogenomics connects somatic mutations to signalling in breast cancer

P Mertins, DR Mani, KV Ruggles, MA Gillette… - Nature, 2016‏ - nature.com
Somatic mutations have been extensively characterized in breast cancer, but the effects of
these genetic alterations on the proteomic landscape remain poorly understood. Here we …

Distinct functions of AKT isoforms in breast cancer: a comprehensive review

N Hinz, M Jücker - Cell Communication and Signaling, 2019‏ - Springer
Background AKT, also known as protein kinase B, is a key element of the PI3K/AKT
signaling pathway. Moreover, AKT regulates the hallmarks of cancer, eg tumor growth …

Buparlisib plus fulvestrant in postmenopausal women with hormone-receptor-positive, HER2-negative, advanced breast cancer progressing on or after mTOR …

A Di Leo, S Johnston, KS Lee, E Ciruelos… - The Lancet …, 2018‏ - thelancet.com
Background Activation of the PI3K/AKT/mTOR pathway occurs frequently in breast cancer
that is resistant to endocrine therapy. Approved mTOR inhibitors effectively inhibit cell …

PI3K/AKT/mTOR: role in breast cancer progression, drug resistance, and treatment

A Guerrero-Zotano, IA Mayer, CL Arteaga - Cancer and Metastasis …, 2016‏ - Springer
Anti-cancer cancer-targeted therapies are designed to exploit a particular vulnerability in the
tumor, which in most cases results from its dependence on an oncogene and/or loss of a …

The PI3K/AKT pathway as a target for cancer treatment

IA Mayer, CL Arteaga - Annual review of medicine, 2016‏ - annualreviews.org
Anticancer targeted therapies are designed to exploit a particular vulnerability in the tumor,
which in most cases results from its dependence on an oncogene and/or loss of a tumor …

[HTML][HTML] The Hippo transducer TAZ confers cancer stem cell-related traits on breast cancer cells

M Cordenonsi, F Zanconato, L Azzolin, M Forcato… - Cell, 2011‏ - cell.com
Cancer stem cells (CSCs) are proposed to drive tumor initiation and progression. Yet, our
understanding of the cellular and molecular mechanisms that underlie CSC properties is …

Luminal B breast cancer: molecular characterization, clinical management, and future perspectives

F Ades, D Zardavas, I Bozovic-Spasojevic… - Journal of clinical …, 2014‏ - ascopubs.org
Gene expression profiling has reshaped our understanding of breast cancer by defining and
characterizing four main intrinsic molecular subtypes: human epidermal growth factor …

Endocrine resistance in breast cancer–an overview and update

R Clarke, JJ Tyson, JM Dixon - Molecular and cellular endocrinology, 2015‏ - Elsevier
Tumors that express detectable levels of the product of the ESR1 gene (estrogen receptor-α;
ERα) represent the single largest molecular subtype of breast cancer. More women …