How to enter a bacterium: bacterial porins and the permeation of antibiotics

JD Prajapati, U Kleinekathöfer… - Chemical …, 2021 - ACS Publications
Despite tremendous successes in the field of antibiotic discovery seen in the previous
century, infectious diseases have remained a leading cause of death. More specifically …

Plant-based phytochemicals as possible alternative to antibiotics in combating bacterial drug resistance

HMA AlSheikh, I Sultan, V Kumar, IA Rather… - Antibiotics, 2020 - mdpi.com
The unprecedented use of antibiotics that led to development of resistance affect human
health worldwide. Prescription of antibiotics imprudently and irrationally in different diseases …

Defining new chemical space for drug penetration into Gram-negative bacteria

S Zhao, JW Adamiak, V Bonifay, J Mehla… - Nature chemical …, 2020 - nature.com
We live in the era of antibiotic resistance, and this problem will progressively worsen if no
new solutions emerge. In particular, Gram-negative pathogens present both biological and …

Membrane-targeting amphiphilic AIE photosensitizer for broad-spectrum bacteria imaging and photodynamic killing of bacteria

H Zhang, C He, L Shen, W Tao, J Zhu, J Song… - Chinese Chemical …, 2023 - Elsevier
An amphiphilic AIE photosensitizer has been successfully developed, which allows for
easily inserting into the bacterial membranes. Binding experiments with phospholipid …

Fast bacterial growth reduces antibiotic accumulation and efficacy

U Łapińska, M Voliotis, KK Lee, A Campey, MRL Stone… - Elife, 2022 - elifesciences.org
Phenotypic variations between individual microbial cells play a key role in the resistance of
microbial pathogens to pharmacotherapies. Nevertheless, little is known about cell …

Development of a universal fluorescent probe for gram‐positive bacteria

HY Kwon, X Liu, EG Choi, JY Lee… - Angewandte Chemie …, 2019 - Wiley Online Library
The rapid and sensitive classification of bacteria is the first step of bacterial community
research and the treatment of infection. Herein, a fluorescent probe BacGO is presented …

Single-cell microfluidics facilitates the rapid quantification of antibiotic accumulation in Gram-negative bacteria

J Cama, M Voliotis, J Metz, A Smith, J Iannucci… - Lab on a Chip, 2020 - pubs.rsc.org
The double-membrane cell envelope of Gram-negative bacteria is a formidable barrier to
intracellular antibiotic accumulation. A quantitative understanding of antibiotic transport in …

Bacterial response mechanism during biofilm growth on different metal material substrates: EPS characteristics, oxidative stress and molecular regulatory network …

J Wang, G Li, H Yin, T An - Environmental research, 2020 - Elsevier
Overwhelming growth of bacterial biofilms on different metal-based pipeline materials are
intractable and pose a serious threat to public health when tap water flows though these …

Synthesis of vancomycin fluorescent probes that retain antimicrobial activity, identify Gram-positive bacteria, and detect Gram-negative outer membrane damage

B Zhang, W Phetsang, MRL Stone, S Kc… - Communications …, 2023 - nature.com
Antimicrobial resistance is an urgent threat to human health, and new antibacterial drugs are
desperately needed, as are research tools to aid in their discovery and development …

Breaching the barrier: quantifying antibiotic permeability across gram-negative bacterial membranes

J Cama, AM Henney, M Winterhalter - Journal of Molecular Biology, 2019 - Elsevier
The double-membrane cell envelope of Gram-negative bacteria is a sophisticated barrier
that facilitates the uptake of nutrients and protects the organism from toxic compounds. An …