[HTML][HTML] Mechanochemistry: A green approach in the preparation of pharmaceutical cocrystals

M Solares-Briones, G Coyote-Dotor, JC Páez-Franco… - Pharmaceutics, 2021‏ - mdpi.com
Mechanochemistry is considered an alternative attractive greener approach to prepare
diverse molecular compounds and has become an important synthetic tool in different fields …

Challenges and opportunities of pharmaceutical cocrystals: a focused review on non-steroidal anti-inflammatory drugs

U Garg, Y Azim - RSC medicinal chemistry, 2021‏ - pubs.rsc.org
The focus of the review is to discuss the relevant and essential aspects of pharmaceutical
cocrystals in both academia and industry with an emphasis on non-steroidal anti …

Design and synthesis of isoniazid-based pyrazolines as potential inhibitors of Mycobacterium tuberculosis with promising radical scavenging action: in-vitro and in …

J Rasgania, R Gavadia, M Varma-Basil… - Journal of Molecular …, 2024‏ - Elsevier
In view of the devastating tuberculosis infections and emerging resistance against available
drugs, novel 5-phenyl-3-(thiophen-2-yl)-4, 5-dihydro-1H-pyrazol-1-yl)(pyridin-4-yl) …

Synthesis, characterization, antimicrobial and antibiofilm activity, and molecular docking analysis of NHC precursors and their Ag-NHC complexes

E Üstün, N Şahin, C Çelik, U Tutar, N Özdemir… - Dalton …, 2021‏ - pubs.rsc.org
Microorganisms attach to surfaces and interfaces and form biofilms which create a sheltered
area for host cell response. Therefore, biofilms provide troubles in fields such as medicine …

Facile synthesis, pharmacological and In silico analysis of succinimide derivatives: An approach towards drug discovery

J Rasgania, R Gavadia, K Jakhar - Journal of Molecular Structure, 2023‏ - Elsevier
The hybrid heterocyclic scaffolds possess extensive medicinal values and significant
pharmaceutical usage. A series of N-substituted-2, 5-dioxopyrrolidine carboxamides …

Design, synthesis and exploration of novel triazinoindoles as potent quorum-sensing inhibitors and radical quenchers

J Rasgania, R Gavadia, N Sahu, P Sharma… - Future Medicinal …, 2024‏ - Taylor & Francis
Background: Antimicrobial resistance has become a critical health concern, and quorum-
sensing exacerbates the resistance by facilitating cell-to-cell communication within the …

Antimicrobial activity, inhibition of biofilm formation, and molecular docking study of novel Ag-NHC complexes

N Şahin, E Üstün, U Tutar, C Celik, N Gürbüz… - Journal of …, 2021‏ - Elsevier
In this study, we reported the synthesis of a new series of Silver (I)-N-heterocyclic carbene
complexes which were obtained from the corresponding new N-heterocyclic carbene (NHC) …

Design and synthesis of triazole-functionalized isatin hybrids with potent anti-proliferative action against triple-negative breast cancer MDA-MB-231 cell line: a hybrid …

J Rasgania, R Gavadia, S Nimesh, L Loveleen… - Journal of the Iranian …, 2024‏ - Springer
Abstract Differently substituted novel 1-(2-((aryl-4 H-1, 2, 4-triazol-3-yl) thio) acetyl) indoline-
2, 3-diones have been synthesized, geometrically optimized, and examined for global …

'Charge Reverse'Halogen Bonding Contacts in Metal-Organic Multi-Component Compounds: Antiproliferative Evaluation and Theoretical Studies

S Banik, T Baishya, RM Gomila, A Frontera… - Inorganics, 2024‏ - mdpi.com
Two new metal–organic multi-component compounds of Ni (II) and Co (II), viz.[Ni (3-CNpy) 2
(H2O) 4] ADS· 2.75 H2O (1) and [Co (3-CNpy) 2 (H2O) 4](4-ClbzSO3) 2 (2)(3-CNpy= 3 …

In acid-aminopyrimidine continuum: experimental and computational studies of furan tetracarboxylate-2-aminopyrimidinium salt

U Garg, Y Azim, M Alam - RSC advances, 2021‏ - pubs.rsc.org
Salts and cocrystals are the two important solid forms when a carboxylic acid crystallizes
with an aminopyrimidine base such that the extent of proton transfer distinguishes between …