Endoplasmic reticulum stress and unfolded protein response in neurodegenerative diseases

R Ghemrawi, M Khair - International journal of molecular sciences, 2020 - mdpi.com
The endoplasmic reticulum (ER) is an important organelle involved in protein quality control
and cellular homeostasis. The accumulation of unfolded proteins leads to an ER stress …

The structure, activation and signaling of IRE1 and its role in determining cell fate

N Siwecka, W Rozpędek-Kamińska, A Wawrzynkiewicz… - Biomedicines, 2021 - mdpi.com
Inositol-requiring enzyme type 1 (IRE1) is a serine/threonine kinase acting as one of three
branches of the Unfolded Protein Response (UPR) signaling pathway, which is activated …

Living dangerously: protective and harmful ER stress responses in pancreatic β-cells

RB Sharma, HV Landa-Galván, LC Alonso - Diabetes, 2021 - Am Diabetes Assoc
Type 2 diabetes (T2D) is a growing cause of poor health, psychosocial burden, and
economic costs worldwide. The pancreatic β-cell is a cornerstone of metabolic physiology …

Peptidomimetic‐based identification of FDA‐approved compounds inhibiting IRE1 activity

D Doultsinos, A Carlesso, C Chintha… - The FEBS …, 2021 - Wiley Online Library
Inositol‐requiring enzyme 1 (IRE1) is a bifunctional serine/threonine kinase and
endoribonuclease that is a major mediator of the unfolded protein response (UPR) during …

Chronic obstructive pulmonary disease and emerging ER stress-related therapeutic targets

JW Yeap, IAH Ali, B Ibrahim, ML Tan - Pulmonary Pharmacology & …, 2023 - Elsevier
COPD pathogenesis is frequently associated with endoplasmic reticulum stress (ER stress)
progression. Targeting the major unfolded protein response (UPR) branches in the ER …

The IRE1 inhibitor Kira6 curtails the inflammatory trait of immunogenic anticancer treatments by targeting Hsp60 independent Of IRE1

R Nicole, K Dimitris, VE Sofie, R Derua, AD Garg… - bioRxiv, 2020 - biorxiv.org
Cellular stress evoked by immunogenic anticancer treatments engaging the unfolded
protein response (UPR) can elicit inflammation with conflicting therapeutic outcomes. To …

Endoplasmic Reticulum Stress and Emerging Therapeutic Targets in Cancer

JW Yeap, ML Tan - Handbook of Cancer and Immunology, 2023 - Springer
Endoplasmic reticulum stress (ER stress) is characterized by the accumulation of misfolded
and unfolded proteins in the ER lumen. To mitigate the imbalanced ER protein-folding …

Unfolded Protein Response Activation Enhances Lung Endothelial Barrier Function

KT Kubra - 2023 - search.proquest.com
The unfolded protein response (UPR) is a homeostatic feedback mechanism that enables
the cells to control endoplasmic reticulum (ER) stress. UPR restores proteostasis by …

[BOOK][B] Exploring NADPH levels during ER stress using novel homoFRET sensors

A Bennett - 2020 - search.proquest.com
In beta-cells, insulin misfolding occurs at rates as high as 20%. Misfolded insulin aggregates
lead to endoplasmic reticulum (ER) stress and the unfolded protein response (UPR). The …

Characterisation of the unfolded protein response in prostate cancer, and investigation of the ATF6 interactome using a modified mammalian expression system.

AM Isac - 2022 - repository.essex.ac.uk
Prostate cancer (PCa) cells grow in an environment which is known to cause endoplasmic
reticulum (ER) stress. This activates a process called the unfolded protein response (UPR) …