Proteasome inhibitors for the treatment of multiple myeloma

S Ito - Cancers, 2020 - mdpi.com
Use of proteasome inhibitors (PIs) has been the therapeutic backbone of myeloma treatment
over the past decade. Many PIs are being developed and evaluated in the preclinical and …

[HTML][HTML] Metformin beyond an anti-diabetic agent: A comprehensive and mechanistic review on its effects against natural and chemical toxins

A Malaekeh-Nikouei, S Shokri-Naei… - Biomedicine & …, 2023 - Elsevier
In addition to the anti-diabetic effect of metformin, a growing number of studies have shown
that metformin has some exciting properties, such as anti-oxidative capabilities, anticancer …

Cardiovascular Toxicity of Proteasome Inhibitors: Underlying Mechanisms and Management Strategies: JACC: CardioOncology State-of-the-Art Review

G Georgiopoulos, N Makris, A Laina, F Theodorakakou… - Cardio Oncology, 2023 - jacc.org
Proteasome inhibitors (PIs) are the backbone of combination treatments for patients with
multiple myeloma and AL amyloidosis, while also indicated in Waldenström's …

Carfilzomib: a promising proteasome inhibitor for the treatment of relapsed and refractory multiple myeloma

SPE Jayaweera… - Frontiers in …, 2021 - frontiersin.org
The proteasome is crucial for the degradation of intracellular proteins and plays an important
role in mediating a number of cell survival and progression events by controlling the levels …

Proteasome inhibitor-related cardiotoxicity: mechanisms, diagnosis, and management

P Wu, O Oren, MA Gertz, EH Yang - Current oncology reports, 2020 - Springer
Abstract Purpose of Review Multiple myeloma is the second most common hematologic
malignancy in the USA, with over 32,000 new cases and nearly 13,000 deaths expected in …

Cardiotoxicity of anticancer drugs: molecular mechanisms, clinical management and innovative treatment

F Gao, T Xu, F Zang, Y Luo, D Pan - Drug Design, Development …, 2024 - Taylor & Francis
With the continuous refinement of therapeutic measures, the survival rate of tumor patients
has been improving year by year, while cardiovascular complications related to cancer …

Canagliflozin mitigates carfilzomib-induced endothelial apoptosis via an AMPK-dependent pathway

MS Dabour, IY Abdelgawad, MKO Grant… - Biomedicine & …, 2023 - Elsevier
Carfilzomib (CFZ) is a proteasome inhibitor approved for relapsed/refractory multiple
myeloma (MM) but its clinical use is limited by cardiovascular toxicity. The mechanisms of …

Cardiovascular toxicity of proteasome inhibitors in multiple myeloma therapy

Y Zheng, S Huang, B **e, N Zhang, Z Liu, G Tse… - Current problems in …, 2023 - Elsevier
The treatment for multiple myeloma has advanced significantly over the past few decades.
Proteasome inhibitors have become the cornerstone of the treatment of multiple myeloma …

Heart failure with targeted cancer therapies: mechanisms and cardioprotection

VS Hahn, KW Zhang, L Sun, V Narayan… - Circulation …, 2021 - Am Heart Assoc
Oncology has seen growing use of newly developed targeted therapies. Although this has
resulted in dramatic improvements in progression-free and overall survival, challenges in …

Obesity and multiple myeloma: Emerging mechanisms and perspectives

A Tentolouris, I Ntanasis-Stathopoulos… - Seminars in Cancer …, 2023 - Elsevier
Obesity is a global pandemic that has been associated with the development of breast,
endometrial, large intestine, renal, esophageal, and pancreatic cancer. Obesity is also …