Design and structural validation of peptide–drug conjugate ligands of the kappa-opioid receptor

E Muratspahić, K Deibler, J Han, N Tomašević… - Nature …, 2023 - nature.com
Despite the increasing number of GPCR structures and recent advances in peptide design,
the development of efficient technologies allowing rational design of high-affinity peptide …

Mind the gap—deciphering GPCR pharmacology using 3D pharmacophores and artificial intelligence

T Noonan, K Denzinger, V Talagayev, Y Chen, K Puls… - Pharmaceuticals, 2022 - mdpi.com
G protein-coupled receptors (GPCRs) are amongst the most pharmaceutically relevant and
well-studied protein targets, yet unanswered questions in the field leave significant gaps in …

Recent Advances in the Synthesis and Applications of m-Aryloxy Phenols

D Amankulova, G Berganayeva, B Kudaibergenova… - Molecules, 2023 - mdpi.com
Since phenol derivatives have high potential as building blocks for the synthesis of bioactive
natural products and conducting polymers, many synthesis methods have been invented. In …

Multi-level biological network analysis and drug repurposing based on leukocyte transcriptomics in severe COVID-19: in silico systems biology to precision medicine

P Sagulkoo, H Chuntakaruk, T Rungrotmongkol… - Journal of personalized …, 2022 - mdpi.com
The coronavirus disease 2019 (COVID-19) pandemic causes many morbidity and mortality
cases. Despite several developed vaccines and antiviral therapies, some patients …

Identificación de posibles dianas terapéuticas en Alzheimer utilizando pipeline bioinformático combinado para aplicarlas al diseño de fármacos asistidos por …

LL Barriga Sanchez - 2023 - repositorio.uta.edu.ec
El acoplamiento molecular demostró que Estradiol y Tricostatina A pueden generar una
inhibición de la proteína CCND1, mientras que Dorsomorfina induce la inhibición de CDK6 …

[ЦИТИРОВАНИЕ][C] Magic™ In Vitro Cell-based Opioid Receptor Functional Assay Service

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