Synthesis, characterization, mechanistic study, in-vitro and in-silico evaluation of antibacterial and antioxidant activities of novel pyrazole-pyrazoline hybrid systems

N Barghady, M Chalkha, I Yamari, N Aflak… - Journal of Molecular …, 2024 - Elsevier
This study describes the synthesis, characterization, and in vitro as well as in silico
assessment of the biological activity of a new series of hybrid molecules. These target …

[HTML][HTML] Efficient Synthesis, Structural Characterization, Antibacterial Assessment, ADME-Tox Analysis, Molecular Docking and Molecular Dynamics Simulations of …

A Arzine, H Hadni, K Boujdi, K Chebbac, N Barghady… - Molecules, 2024 - mdpi.com
This work describes the synthesis, characterization, and in vitro and in silico evaluation of
the biological activity of new functionalized isoxazole derivatives. The structures of all new …

Insights into the inhibitory potential of novel hydrazinyl thiazole-linked indenoquinoxaline against alpha-amylase: a comprehensive QSAR, pharmacokinetic, and …

O Abchir, I Yamari, AM Shtaiwi, H Nour… - Journal of …, 2024 - Taylor & Francis
The rising prevalence of diabetes necessitates the development of novel drugs, especially
given the side effects associated with current medications like Acarbose and Voglibose. A …

Synthesis, antifungal evaluation, two‐dimensional quantitative structure–activity relationship and molecular docking studies of isoxazole derivatives as potential …

K Tripathi, P Kaushik, DK Yadav… - Pest Management …, 2024 - Wiley Online Library
BACKGROUND Sheath blight and bakanae disease, prominent among emerging rice
ailments, exert a profound impact on rice productivity, causing severe impediments to crop …

An investigation of the adsorption of Congo red dye on two naturally occurring adsorbents Hydroxyapatite and Bentonite: An Experimental Analysis, DFT calculations …

A Grouli, A Chraka, Y Bachra, M Elkouali, S Chtita… - Heliyon, 2024 - cell.com
Congo Red (CR) dye is classified as a toxic and carcinogenic substance, posing significant
health and environmental risks. To address this issue, the adsorption efficiency of CR on …

Michael addition of ethyl acetoacetate on dibenzylideneacetone derivatives: Synthesis, spectroscopy, antimicrobial and in silico studies

A Mouhib, B Es-Sounni, M Laghmari, J Touhtouh… - Journal of Molecular …, 2025 - Elsevier
A series of trisubstituted cyclohexenones incorporating a styryl framework were synthesized
by Michael addition reaction of ethyl acetoacetate onto dibenzylideneacetone derivatives …

Antimicrobial activity of isoxazole derivatives: A brief overview

K Vashisht, P Sethi, A Bansal… - Vietnam Journal of …, 2024 - Wiley Online Library
Due to their extensive range of biological actions, isoxazole and its analogues stand out
among other heterocyclic compounds as a very important class of heterocycles. Over recent …

[HTML][HTML] New Quinazolin-4 (3H)-One Derivatives Incorporating Isoxazole Moiety as Antioxidant Agents: Synthesis, Structural Characterization, and Theoretical DFT …

Y Rhazi, R Sghyar, N Deak, B Es-Sounni, B Rossafi… - Pharmaceuticals, 2024 - mdpi.com
Background: This research centers on the development and spectroscopic characterization
of new quinazolin-4 (3H)-one-isoxazole derivatives (5a–e). The aim was to investigate the …

Deciphering the cytotoxic and antioxidant potential of 3, 5-disubstituted isoxazole-linked benzimidazolone derivatives

M Adardour, S Drioua, MA Lahcen, I Hdoufane… - Journal of Molecular …, 2025 - Elsevier
A series of new isoxazole derivatives containing a benzimidazolone has been synthesized
by cycloaddition reaction using various nitrile oxides. In all cases, these cycloadditions are …

Reactivity of (3‐(4‐Fluorophenyl) oxyran‐2‐yl)(naphthalene‐2‐yl) methanone Toward Some Nucleophiles for Preparing Promising Agents with Antimicrobial and …

HS Khalaf, ER Kotb, NAM Abdelwahed… - …, 2024 - Wiley Online Library
Abstract (3‐(4‐Fluorophenyl) oxyran‐2‐yl)(naphthalene‐2‐yl) methanone 2 was prepared
from the reaction of 3‐(4‐fluorophenyl)‐1‐(naphthalen‐2‐yl) prop‐2‐en‐1‐one (1) with …