Privileged scaffolds as starting points toward biologically active molecules represent a
neuralgic point in drug discovery. The ability of synthetic chemists concerned with their …

Pyrazoline core is a very interesting five‐membered heterocycle, which has been explored
in recent years due to its vast applications as the core structure of bioactive and industrial …

In continuation of our study of novel quinolines with anti-inflammatory activity using the
Pfitzinger reaction, several new quinoline derivatives were synthesized and tested for their …

A highly regioselective cycloaddition procedure of electron-deficient allenes with
trifluorodiazoethane (CF3CHN2) is described. In absence of bases, the reaction proceeded …

The first catalytic enantioselective iodoaminocyclization of β, γ-unsaturated hydrazones has
been developed with the help of a trans-1, 2-diaminocyclohexane-derived bifunctional …

A general catalytic methodology for the synthesis of pyrazolines from α‐diazo compounds
and conjugated alkenes is reported. The direct hydrogen atom transfer (HAT) process of α …

Antitumor activity using 59 cancer cell lines and enzyme inhibitory activity of a newly
synthesized pyrazoline-linked 4-methylsulfonylphenyl scaffold (compounds 18a–q) were …

A simple, efficient, and environment friendly protocol for the synthesis of 1, 3, 5-
triarylpyrazoles and 1, 3, 5-triarylpyrazolines in [bmim][PF6] ionic liquid mediated by Cu …

Generation of C2F5CHN2 In Situ and Its First Reaction: [3+2] Cycloaddition with Alkenes -
Mykhailiuk - 2014 - Chemistry – A European Journal - Wiley Online Library Skip to Article Content …

New thiazolylmethoxyphenyl pyrimidines (7a–g) have been conveniently synthesized with
better yields by cyclocondensing 3-(4-((2-phenylthiazol-4-yl) methoxy) phenyl)-1-(4 …