Allosteric SHP2 inhibitors in cancer: Targeting the intersection of RAS, resistance, and the immune microenvironment

DL Kerr, F Haderk, TG Bivona - Current opinion in chemical biology, 2021 - Elsevier
The nonreceptor protein tyrosine phosphatase SHP2 (encoded by PTPN11) integrates
growth and differentiation signals from receptor tyrosine kinases (RTKs) into the …

Functions of Shp2 in cancer

J Zhang, F Zhang, R Niu - Journal of cellular and molecular …, 2015 - Wiley Online Library
Diagnostics and therapies have shown evident advances. Tumour surgery, chemotherapy
and radiotherapy are the main techniques in treat cancers. Targeted therapy and drug …

SHP2 sails from physiology to pathology

M Tajan, A de Rocca Serra, P Valet, T Edouard… - European journal of …, 2015 - Elsevier
Over the two past decades, mutations of the PTPN11 gene, encoding the ubiquitous protein
tyrosine phosphatase SHP2 (SH2 domain-containing tyrosine phosphatase 2), have been …

Reactive oxygen species and mitochondrial homeostasis as regulators of stem cell fate and function

DQ Tan, T Suda - Antioxidants & redox signaling, 2018 - liebertpub.com
Significance: The precise role and impact of reactive oxygen species (ROS) in stem cells,
which are essential for lifelong tissue homeostasis and regeneration, remain of significant …

Correlation of mutation profile and response in patients with myelofibrosis treated with ruxolitinib

KP Patel, KJ Newberry, R Luthra… - Blood, The Journal …, 2015 - ashpublications.org
Although most patients with myelofibrosis (MF) derive benefit from ruxolitinib, some are
refractory, have a suboptimal response, or quickly lose their response. To identify genes that …

[PDF][PDF] Shp2 promotes liver cancer stem cell expansion by augmenting β‐catenin signaling and predicts chemotherapeutic response of patients

D ** tissue macrophage populations
R Paccoud, C Saint-Laurent, E Piccolo… - Science Translational …, 2021 - science.org
Insulin resistance is a key event in type 2 diabetes onset and a major comorbidity of obesity.
It results from a combination of fat excess–triggered defects, including lipotoxicity and …

Dynamics of thymus function and T cell receptor repertoire breadth in health and disease

D Granadier, L Iovino, S Kinsella… - Seminars in …, 2021 - Springer
T cell recognition of unknown antigens relies on the tremendous diversity of the T cell
receptor (TCR) repertoire; generation of which can only occur in the thymus. TCR repertoire …