[HTML][HTML] Impact of regional differences along the gastrointestinal tract of healthy adults on oral drug absorption: An UNGAP review

M Vertzoni, P Augustijns, M Grimm, M Koziolek… - European journal of …, 2019 - Elsevier
Oral administration is the most common route of drug delivery. The absorption of a drug from
the gut into the bloodstream involves disintegration of the solid dosage form, dissolution of …

Application of targeted mass spectrometry in bottom-up proteomics for systems biology research

NP Manes, A Nita-Lazar - Journal of proteomics, 2018 - Elsevier
The enormous diversity of proteoforms produces tremendous complexity within cellular
proteomes, facilitates intricate networks of molecular interactions, and constitutes a …

Non-uniformity of changes in drug-metabolizing enzymes and transporters in liver cirrhosis: implications for drug dosage adjustment

E El-Khateeb, B Achour, ZM Al-Majdoub… - Molecular …, 2021 - ACS Publications
Liver cirrhosis is a chronic disease that affects the liver structure, protein expression, and
overall metabolic function. Abundance data for drug-metabolizing enzymes and transporters …

Large‐scale multiplex absolute protein quantification of drug‐metabolizing enzymes and transporters in human intestine, liver, and kidney microsomes by SWATH‐MS …

K Nakamura, M Hirayama‐Kurogi, S Ito, T Kuno… - …, 2016 - Wiley Online Library
The purpose of the present study was to examine simultaneously the absolute protein
amounts of 152 membrane and membrane‐associated proteins, including 30 metabolizing …

Quantitative proteomics of clinically relevant drug-metabolizing enzymes and drug transporters and their intercorrelations in the human small intestine

N Couto, ZM Al-Majdoub, S Gibson, PJ Davies… - Drug Metabolism and …, 2020 - Elsevier
The levels of drug-metabolizing enzymes (DMEs) and transporter proteins in the human
intestine are pertinent to determine oral drug bioavailability. Despite the paucity of reports on …

Oral drug absorption in pediatrics: the intestinal wall, its developmental changes and current tools for predictions

JM Nicolas, F Bouzom, C Hugues… - … & drug disposition, 2017 - Wiley Online Library
The dissolution, intestinal absorption and presystemic metabolism of a drug depend on its
physicochemical characteristics but also on numerous physiological (eg gastrointestinal pH …

Regional expression levels of drug transporters and metabolizing enzymes along the pig and human intestinal tract and comparison with Caco-2 cells

SFC Vaessen, MMH van Lipzig, RHH Pieters… - Drug metabolism and …, 2017 - Elsevier
Intestinal transporter proteins and metabolizing enzymes play a crucial role in the oral
absorption of a wide variety of drugs. The aim of the current study was to characterize better …

Identification and quantification of blood–brain barrier transporters in isolated rat brain microvessels

H Al Feteisi, ZM Al‐Majdoub, B Achour… - Journal of …, 2018 - Wiley Online Library
The blood–brain barrier (BBB) maintains brain homeostasis by tightly regulating the
exchange of molecules with systemic circulation. It consists primarily of microvascular …

Quantitative atlas of cytochrome P450, UDP-glucuronosyltransferase, and transporter proteins in jejunum of morbidly obese subjects

E Miyauchi, M Tachikawa, X Declèves… - Molecular …, 2016 - ACS Publications
Protein expression levels of drug-metabolizing enzymes and transporters in human jejunal
tissues excised from morbidly obese subjects during gastric bypass surgery were evaluated …

Critical issues and optimized practices in quantification of protein abundance level to determine interindividual variability in DMET proteins by LC‐MS/MS proteomics

DK Bhatt, B Prasad - Clinical Pharmacology & Therapeutics, 2018 - Wiley Online Library
Protein quantification data on drug metabolizing enzymes and transporters (collectively
referred as DMET proteins) in human tissues are useful in predicting interindividual …