Benzothiazole (BTA) and its derivatives are the most important heterocyclic compounds,
which are common and integral feature of a variety of natural products and pharmaceutical …

Heterocycles bearing nitrogen, sulphur and thiazole moieties constitute the core structure of
a number of biologically interesting compounds. Benzothiazole, a group of xenobiotic …

A new, convenient method for the syntheses of 2-substituted benzimidazole and
benzothizole is described. Short reaction times, large-scale synthesis, easy and quick …

A series of water-soluble l-lysyl-and l-alanyl-amide prodrugs of the lipophilic antitumor 2-(4-
aminophenyl) benzothiazoles has been synthesized to address formulation and …

Benzothiazole is an organic compound bearing a heterocyclic nucleus (thiazole) which
imparts a broad spectrum of biological activities to it. The significant and potent activity of …

Synthetic routes to a series of mono-and difluorinated 2-(4-amino-3-substituted-phenyl)
benzothiazoles have been devised. Whereas mixtures of regioisomeric 5-and 7-fluoro …

Phthalic anhydride is a highly toxic substance, facing, however, the problem of hydrolysis. In
fact, it is rapidly hydrolyzed in aqueous medium, generating phthalic acid as the final …

2-(4-Aminophenyl) benzothiazoles 1 and their N-acetylated forms have been converted to C-
and N-hydroxylated derivatives to investigate the role of metabolic oxidation in the mode of …

Sažetak A series of new benzothiazole derivatives 6a-h have been synthesized, in five
steps, from substituted phenols via the 1, 3, 4-oxadiazole-2-thiones 5a-h. The in vitro …

The Pd-and Cu-mediated reaction of a large variety of π-electron sufficient heteroarenes,
which include free (NH)-imidazoles,-benzimidazole and-indole, with aryl iodides under …