Inhibition of FGF‐FGFR and VEGF‐VEGFR signalling in cancer treatment

G Liu, T Chen, Z Ding, Y Wang, Y Wei, X Wei - Cell proliferation, 2021 - Wiley Online Library
The sites of targeted therapy are limited and need to be expanded. The FGF‐FGFR
signalling plays pivotal roles in the oncogenic process, and FGF/FGFR inhibitors are a …

Molecular hybrids: A five-year survey on structures of multiple targeted hybrids of protein kinase inhibitors for cancer therapy

OM Soltan, ME Shoman, SA Abdel-Aziz… - European Journal of …, 2021 - Elsevier
Protein kinases have grown over the past few years as a crucial target for different cancer
types. With the multifactorial nature of cancer, and the fast development of drug resistance …

Fibroblast growth factor receptors (FGFRs) and noncanonical partners in cancer signaling

HR Ferguson, MP Smith, C Francavilla - Cells, 2021 - mdpi.com
Increasing evidence indicates that success of targeted therapies in the treatment of cancer is
context-dependent and is influenced by a complex crosstalk between signaling pathways …

Research progress on the PI3K/AKT signaling pathway in gynecological cancer

X Shi, J Wang, Y Lei, C Cong… - Molecular medicine …, 2019 - spandidos-publications.com
Abstract The phosphatidylinositol 3‑kinase (PI3K)/protein kinase B (AKT) signaling pathway
is involved in the regulation of multiple cellular physiological processes by activating …

Silencing of hsa_circ_0009035 suppresses cervical cancer progression and enhances radiosensitivity through microRNA 889-3p-dependent regulation of HOXB7

X Zhao, W Dong, G Luo, J **e, J Liu… - Molecular and Cellular …, 2021 - Taylor & Francis
Circular RNAs (circRNAs), a novel type of endogenous noncoding RNAs, have been
identified as critical regulators in human carcinogenesis. Here, we investigated the precise …

Design, synthesis, and anticancer evaluation of novel quinoline derivatives of ursolic acid with hydrazide, oxadiazole, and thiadiazole moieties as potent MEK …

XY **, H Chen, DD Li, AL Li, WY Wang… - Journal of enzyme …, 2019 - Taylor & Francis
In this article, a series of novel quinoline derivatives of ursolic acid (UA) bearing hydrazide,
oxadiazole, or thiadiazole moieties were designed, synthesised, and screened for their in …

Genomic landscapes of EBV-associated nasopharyngeal carcinoma vs. HPV-associated head and neck cancer

HL Ngan, L Wang, KW Lo, VWY Lui - Cancers, 2018 - mdpi.com
Epstein-Barr virus-positive nasopharyngeal carcinoma (EBV (+) NPC), and human
papillomavirus-positive head and neck squamous cell carcinoma (HPV (+) HNSCC) are two …

Targeted therapy with PI3K and FGFR inhibitors on human papillomavirus positive and negative tonsillar and base of tongue cancer lines with and without …

S Holzhauser, N Wild, M Zupancic, RG Ursu… - Frontiers in …, 2021 - frontiersin.org
Objectives Human papillomavirus positive (HPV+) tonsillar and base of tongue squamous
cell carcinoma (TSCC/BOTSCC), the major subsites of oropharyngeal squamous cell …

XCL1 expression correlates with CD8-positive T cells infiltration and PD-L1 expression in squamous cell carcinoma arising from mature cystic teratoma of the ovary

R Tamura, K Yoshihara, H Nakaoka, N Yachida… - Oncogene, 2020 - nature.com
Molecular characteristics of carcinoma arising from mature cystic teratoma of the ovary
(MCT) remain unclear due to its rarity. We analyzed RNA-sequencing data of 2322 pan …

Targeting fibroblast growth factor receptor (FGFR) and phosphoinositide 3-kinase (PI3K) signaling pathways in medulloblastoma cell lines

S Holzhauser, M Lukoseviciute, T Andonova… - Anticancer …, 2020 - ar.iiarjournals.org
Background/Aim: Medulloblastoma (MB) accounts for~ 20% of pediatric malignant central
nervous system tumors. Treatment strategies, including surgery, radiation therapy and/or …