Natural products and their analogues acting against Mycobacterium tuberculosis: A recent update

G Kumar - Drug Development Research, 2023 - Wiley Online Library
Tuberculosis (TB) remains one of the deadliest infectious diseases caused by
Mycobacterium tuberculosis (M. tb). It is responsible for significant causes of mortality and …

Tryptanthrins as multi-bioactive agents: discovery, diversity distribution and synthesis

K Alam, MS Hossain, Y Zhao, Z Zhang, S Xu, J Hao… - Bioorganic …, 2024 - Elsevier
Tryptanthrin and its derivatives, representing a type of alkaloids with indoloquinazoline
structures, were first obtained from blue plants and indigo, and then extracted from fungi …

Novel Derivatives of Quinoxaline-2-carboxylic Acid 1, 4-Dioxides as Antimycobacterial Agents: Mechanistic Studies and Therapeutic Potential

SG Frolova, AA Vatlin, DA Maslov, B Yusuf… - Pharmaceuticals, 2023 - mdpi.com
The World Health Organization (WHO) reports that tuberculosis (TB) is one of the top 10
leading causes of global mortality. The increasing incidence of multidrug-resistant TB …

The Antitubercular Activities of Natural Products with Fused-Nitrogen-Containing Heterocycles

HI Boshoff, N Malhotra, CE Barry III, S Oh - Pharmaceuticals, 2024 - mdpi.com
Tuberculosis (TB) is notorious as the leading cause of death worldwide due to a single
infectious entity and its causative agent, Mycobacterium tuberculosis (Mtb), has been able to …

Synthesis and characterization of novel 2-acyl-3-trifluoromethylquinoxaline 1, 4-dioxides as potential antimicrobial agents

GI Buravchenko, DA Maslov, MS Alam… - Pharmaceuticals, 2022 - mdpi.com
The emergence of drug resistance in pathogens leads to a loss of effectiveness of
antimicrobials and complicates the treatment of bacterial infections. Quinoxaline 1, 4 …

Polymeric nanoparticles as a promising drug delivery platform for the efficacious delivery of toll-like receptor 7/8 agonists and IDO-inhibitor

J Rathee, A Kaur, R Kanwar, D Kaushik… - Colloids and Surfaces A …, 2022 - Elsevier
The current investigation delineates the poly (lactide-co-glycolic acid) nanoparticles (PLGA
NPs) formulation as the drug encapsulating assembly using nanoprecipitation method …

Recent advances of tryptanthrin and its derivatives as potential anticancer agents

X Zhou - RSC Medicinal Chemistry, 2024 - pubs.rsc.org
Tryptanthrin is one of the well-known natural alkaloids with the broader spectrum of
biological activities as anti-inflammatory, anticancer, antibacterial, antifungal, antiviral …

Repurposing Based Identification of Novel Inhibitors against MmpS5-MmpL5 Efflux Pump of Mycobacterium smegmatis: A Combined In Silico and In Vitro Study

M Shahbaaz, DA Maslov, AA Vatlin, VN Danilenko… - Biomedicines, 2022 - mdpi.com
In the current era of a pandemic, infections of COVID-19 and Tuberculosis (TB) enhance the
detrimental effects of both diseases in suffering individuals. The resistance mechanisms …

Genetic interaction between F‐box motif encoding YDR131C and retrograde signaling‐related RTG1 regulates the stress response and apoptosis in Saccharomyces …

H Shoket, M Pandita, M Sharma… - … of Biochemical and …, 2021 - Wiley Online Library
The retrograde signaling pathway is well conserved from yeast to humans, which regulates
cell adaptation during stress conditions and prevents cell death. One of its components …

Transcriptomic Profile of Mycobacterium smegmatis in Response to an Imidazo[1,2-b][1,2,4,5]tetrazine Reveals Its Possible Impact on Iron Metabolism

AA Vatlin, EA Shitikov, M Shahbaaz… - Frontiers in …, 2021 - frontiersin.org
Tuberculosis (TB), caused by the Mycobacterium tuberculosis complex bacteria, is one of
the most pressing health problems. The development of new drugs and new therapeutic …