Adenosine receptor antagonists: Recent advances and therapeutic perspective

A Saini, R Patel, S Gaba, G Singh, GD Gupta… - European Journal of …, 2022 - Elsevier
Adenosine is an endogenous purine-based nucleoside expressed nearly in all body tissues.
It regulates various body functions by activating four G-protein coupled receptors, A 1, A 2A …

Recent developments in new therapeutic agents against Alzheimer and Parkinson diseases: in-silico approaches

P Cruz-Vicente, LA Passarinha, S Silvestre, E Gallardo - Molecules, 2021 - mdpi.com
Neurodegenerative diseases (ND), including Alzheimer's (AD) and Parkinson's Disease
(PD), are becoming increasingly more common and are recognized as a social problem in …

Methylxanthines and neurodegenerative diseases: an update

D Janitschke, AA Lauer, CM Bachmann, HS Grimm… - Nutrients, 2021 - mdpi.com
Methylxanthines (MTX) are purine derived xanthine derivatives. Whereas naturally occurring
methylxanthines like caffeine, theophylline or theobromine are widely consumed in food …

Recent advances in the biological significance of xanthine and its derivatives: a review

A Kapri, S Pant, N Gupta, S Nain - Pharmaceutical Chemistry Journal, 2022 - Springer
Xanthine is the most ubiquitous heterocyclic aromatic compound and have attracted much
synthetic interest due to their numerous pharmacological activities. It is one of the principal …

Drug Development for Alzheimer's and Parkinson's Disease: Where Do We Go Now?

L Sequeira, S Benfeito, C Fernandes, I Lima, J Peixoto… - Pharmaceutics, 2024 - mdpi.com
Neurodegenerative diseases (NDs) are a set of progressive, chronic, and incurable
diseases characterized by the gradual loss of neurons, culminating in the decline of …

Synthesis, QSAR modeling, and molecular docking of novel fused 7‐deazaxanthine derivatives as adenosine A2A receptor antagonists

LV Muzychka, EV Verves, IO Yaremchuk… - Chemical Biology & …, 2022 - Wiley Online Library
Predictive QSAR models for the search of new adenosine A2A receptor antagonists were
developed by using OCHEM platform. The predictive ability of the regression models has …

Once Upon a Time Adenosine and Its Receptors: Historical Survey and Perspectives as Potential Targets for Therapy in Human Diseases

D Catarzi, F Varano, S Calenda, E Vigiani… - Purinergic Receptors and …, 2023 - Springer
Endogenous autacoid adenosine plays important physiological roles in various tissues and
organs by acting through A1, A2A, A2B, and A3 receptors. Dysregulated extracellular …

Koffein, Schokolade und Adenosin A2A Rezeptorantagonisten in der Behandlung des Parkinson Syndroms

H Reichmann - Fortschritte der Neurologie· Psychiatrie, 2023 - thieme-connect.com
Hintergrund Patienten mit einem idiopathischen Parkinson-Syndrom können offenbar vom
Koffeinkonsum profitieren, wie bereits eine Reihe experimenteller und klinischer Studien …

[ЦИТИРОВАНИЕ][C] Drug Development for Alzheimer's and Parkinson's Disease: Where Do We Go Now? Pharmaceutics 2024, 16, 708

L Sequeira, S Benfeito, C Fernandes, I Lima, J Peixoto… - 2024 - europepmc.org
Neurodegenerative diseases (NDs) are a set of progressive, chronic, and incurable
diseases characterized by the gradual loss of neurons, culminating in the decline of …