It Takes Two to Tango: Directly Optimizing for Constrained Synthesizability in Generative Molecular Design

J Guo, P Schwaller - arxiv preprint arxiv:2410.11527, 2024 - arxiv.org
Constrained synthesizability is an unaddressed challenge in generative molecular design.
In particular, designing molecules satisfying multi-parameter optimization objectives, while …

Active Learning to Select the Most Suitable Reagents and One-Step Organic Chemistry Reactions for Prioritizing Target-Specific Hits from Ultralarge Chemical Spaces

V Kozyrev, F Sindt, D Rognan - Journal of Chemical Information …, 2025 - ACS Publications
Designing chemically novel and synthesizable ligands from the largest possible chemical
space is a major issue in modern drug discovery to identify early hits that are easily …

Neural Genetic Search in Discrete Spaces

H Kim, S Choi, J Son, J Park, C Kwon - arxiv preprint arxiv:2502.10433, 2025 - arxiv.org
Effective search methods are crucial for improving the performance of deep generative
models at test time. In this paper, we introduce a novel test-time search method, Neural …

Procedural Synthesis of Synthesizable Molecules

M Sun, A Lo, M Guo, J Chen, W Matusik… - … Conference on Learning … - openreview.net
Designing synthetically accessible molecules and recommending analogs to
unsynthesizable molecules are important problems for accelerating molecular discovery. We …