In the field of drug discovery, isoxazole is a five-membered heterocyclic moiety commonly
found in many commercially available drugs. In view of their enormous significance, it is …

Abstract β‐Carboline, a privileged scaffold in the alkaloid family, has a broad spectrum of
medicinal properties and is found in several commercial drugs, such as tadalafil …

The involvement of 1, 3-dipolar cycloaddition (1, 3-DP), double bond migration, metathesis,
and nitrile oxide (including in situ-generated nitrile oxide) as dipoles, together with the C= C …

N-arylated heterocycles are a significant class of core scaffolds in medicinal chemistry,
materials science, and agrochemistry, highlighting their importance in various fields. The …

Synthesis of β-carboline based natural products and synthetic derivatives is one of the
frontier areas of research owing to their medicinal properties. It is envisaged that 3-formyl-9H …

A one‐pot strategy for constructing trisubstituted pyridine derivatives had been established
via phosphine‐catalyzed annulation and DDQ oxidative aromatization reactions. This …

Herein, a catalyst‐free method for synthesizing 4, 5‐dihydroisoxazole‐5‐methanols is
proposed, whereby isoxazolines are constructed through the NCS‐mediated 1, 3‐dipolar …

A simple and highly efficient one‐pot, metal‐free approach has been developed for the
synthesis of β‐carboline− pyrazole/− pyrazoline‐based molecular hybrids. The synthesis of …

The functionalized tetrahydrochromeno [4′, 3′: 2, 3] indolizino [8, 7-b] indoles were
conveniently synthesized in high yields by one-pot domino reaction of tryptamines, alkyl …

A robust transition-metal-free strategy is presented to access novel β-carboline-tethered
benzothiophenone derivatives from 1 (3)-formyl-β-carbolines using elemental sulfur …