A review on biological and medicinal significance of thiazoles

PM Jadhav, S Kantevari, AB Tekale… - … , Sulfur, and Silicon …, 2021 - Taylor & Francis
Thiazole, a five-membered heterocyclic compound constitutes the skeleton of various
commercially marketed drug candidates and the heart-core in a diverse range of entities of …

[PDF][PDF] Synthesis and anticancer activities of thiazoles, 1, 3-thiazines, and thiazolidine using chitosan-grafted-poly (vinylpyridine) as basic catalyst

SM Gomha, SM Riyadh, EA Mahmmoud… - …, 2015 - triggered.stanford.clockss.org
Three different series of ethylidenehydrazonothiazoles 5a-c, 6a-c, ethylidenehydrazono-1, 3-
thiazines 9a-i and ethylidenehydrazonothiazolidine 12 have been prepared via reactions of …

L-Proline catalyzed green synthesis and anticancer evaluation of novel bioactive benzil bis-hydrazones under grinding technique

AR Sayed, SM Gomha, HM Abd El-lateef… - … Chemistry Letters and …, 2021 - Taylor & Francis
ABSTRACT L-Proline organocatalyst was investigated as an efficient and environmentally
benign catalyst for synthesis of some novel bioactive benzil bis (2-cyano-3-aryl-2 …

Discovery of thiazole-based-chalcones and 4-hetarylthiazoles as potent anticancer agents: Synthesis, docking study and anticancer activity

TA Farghaly, GS Masaret, ZA Muhammad… - Bioorganic chemistry, 2020 - Elsevier
The crucial need for novel antitumor agents with high selectivity toward cancer cells has
promoted us to synthesize new series of thiazole-based chalcones and 4-hetarylthiazoles …

Synthesis, characterization, and pharmacological evaluation of some novel thiadiazoles and thiazoles incorporating pyrazole moiety as anticancer agents

SM Gomha, TA Salah, AO Abdelhamid - Monatshefte für Chemie …, 2015 - Springer
Abstract Two series of novel 2-[[1-(5-methyl-1-phenyl-5-substituted-1 H-pyrazol-4-yl)
ethylidene] hydrazono]-3-phenyl-2, 3-dihydro-1, 3, 4-thiadiazole derivatives and 2-[5-(4 …

Synthesis and biological evaluation of some novel thiazole-based heterocycles as potential anticancer and antimicrobial agents

S Abu-Melha, MM Edrees, HH Salem, NA Kheder… - Molecules, 2019 - mdpi.com
A novel series of thiazole-based heterocycles was synthesized using 1, 3-dipolar
cycloaddition reactions in the presence of chitosan-grafted-poly (vinylpyridine) as an eco …

Synthesis and Characterization of Some New Bis-Pyrazolyl-Thiazoles Incorporating the Thiophene Moiety as Potent Anti-Tumor Agents

SM Gomha, MM Edrees, FMA Altalbawy - International journal of …, 2016 - mdpi.com
A new series of 1, 4-bis (1-(5-(aryldiazenyl) thiazol-2-yl)-5-(thiophen-2-yl)-4, 5-dihydro-1 H-
pyrazol-3-yl) benzenes 3a–i were synthesized via reaction of 5, 5′-(1, 4-phenylene) bis (3 …

A novel highly crystalline Fe 4 (Fe (CN) 6) 3 concave cube anode material for Li-ion batteries with high capacity and long life

X He, L Tian, M Qiao, J Zhang, W Geng… - Journal of Materials …, 2019 - pubs.rsc.org
Recently, Prussian blue and its analogues (PBs) have been widely investigated as cathode
materials for sodium ion batteries (SIBs), but have rarely been reported as anode materials …

Microwave-assisted one pot three-component synthesis of some novel pyrazole scaffolds as potent anticancer agents

SM Gomha, MM Edrees, RAM Faty… - Chemistry Central …, 2017 - Springer
Abstract Background Pyrazoles, thiazoles and 1, 3, 4-thiadiazoles have been reported to
possess various pharmacological activities. Results An efficient and a novel approach for …

Synthesis, characterization and DFT calculated properties of electron-rich hydrazinylthiazoles: Experimental and computational synergy

H Mehmood, M Khalid, M Haroon, T Akhtar… - Journal of Molecular …, 2021 - Elsevier
Abstract Rare electron-rich 1-(2-{2-[(aryl) methylidene](R-hydrazinyl}-4-methyl-1, 3-thiazol-5-
yl) ethan-1-ones [ArCHdouble bondNN (R) C 3 NS (Me)(COMe); Ar= 2-, 3-or 4-MeOC 6 H 4 …