Recent developments of transition-state analogue glycosidase inhibitors of non-natural product origin

VH Lillelund, HH Jensen, X Liang, M Bols - Chemical reviews, 2002‏ - ACS Publications
Glycosidase inhibitors have been subject to extensive interest in the past decade. As
glycoside cleavage is a biologically widespread process, glycosidase inhibitors have many …

Glycosidase mechanisms

A Vasella, GJ Davies, M Böhm - Current opinion in chemical biology, 2002‏ - Elsevier
The three-dimensional structure of glycosidases and of their complexes and the study of
transition-state mimics reveal structural details that correlate with mechanism. Of particular …

Catalytic mechanism of enzymic glycosyl transfer

ML Sinnott - Chemical Reviews, 1990‏ - ACS Publications
At least in terms of simple tonnage, glycosyl transfer must be accounted one of the most
important biochemical reactions, since around two-thirds of the carbon in the biosphere …

Stereochemistry of nucleophilic substitution reactions depending upon substituent: evidence for electrostatic stabilization of pseudoaxial conformers of oxocarbenium …

L Ayala, CG Lucero, JAC Romero… - Journal of the …, 2003‏ - ACS Publications
Lewis acid-mediated nucleophilic substitution reactions of substituted tetrahydropyran
acetates reveal that the conformational preferences of six-membered-ring cations depend …

Toward a Detailed Understanding of Base Excision Repair Enzymes:  Transition State and Mechanistic Analyses of N-Glycoside Hydrolysis and N-Glycoside …

PJ Berti, JAB McCann - Chemical reviews, 2006‏ - ACS Publications
This review focuses on the chemistry performed by base excision repair (BER) enzymes,
enzymes that remove nucleobases from DNA in the first step of the repair of many types of …

Stereochemical reversal of nucleophilic substitution reactions depending upon substituent: reactions of heteroatom-substituted six-membered-ring oxocarbenium ions …

JAC Romero, SA Tabacco… - Journal of the American …, 2000‏ - ACS Publications
Although conformational preferences of neutral six-memberedring systems are dominated
by steric effects, 1 recent computational studies suggest that electronic effects exert a …

Synthesis and biological activity of natural aminocyclopentitol glycosidase inhibitors: mannostatins, trehazolin, allosamidins, and their analogues

A Berecibar, C Grandjean… - Chemical …, 1999‏ - pubmed.ncbi.nlm.nih.gov
Synthesis and Biological Activity of Natural Aminocyclopentitol Glycosidase Inhibitors:
Mannostatins, Trehazolin, Allosamidins, and Their Analogues Synthesis and Biological …

Antiviral therapy for human immunodeficiency virus infections

E De Clercq - Clinical microbiology reviews, 1995‏ - journals.asm.org
Depending on the stage of their intervention with the viral replicative cycle, human
immunodeficiency virus inhibitors could be divided into the following groups:(i) adsorption …

[ספר][B] C-Glycoside synthesis

M Postema - 2020‏ - taylorfrancis.com
This book examines methods particularly well suited for either a-or bC-glycoside formation. It
helps field workers quickly select the best method for synthesizing a particular type of C …

Enzyme-catalyzed aldol condensation for asymmetric synthesis of azasugars: synthesis, evaluation, and modeling of glycosidase inhibitors

T Kajimoto, KKC Liu, RL Pederson… - Journal of the …, 1991‏ - ACS Publications
A combined fructose 1, 6-diphosphate aldolase reaction and catalytic reductive animation
has been used in the asymmetric synthesis of azasugars structurally correspondingto 7V …