Benzoxazole is an attractive scaffold in medicinal chemistry due to its diverse biological
applications. From 2016 to 2023, a plethora of benzoxazole derivatives have been …

Benzoxazoles and benzothiazoles are a class of aromatic heterocyclic compounds having
similar ring structures, in which a benzene ring is fused to the 4 and 5 positions of the 1, 3 …

An environmentally friendly, versatile multicomponent reaction for synthesizing isoxazol-5-
one and pyrazol-3-one derivatives has been developed, utilizing a freshly prepared g-C3N4 …

Novel benzimidazoles, benzothiazoles, and benzoxazoles linked to N-arylacetamide were
synthesized in good yields by reacting a series of 2-oxo-2-(arylamino) ethyl 4 …

The necessary use of large amounts of a homogeneous electrolyte represents a major issue
and challenge for the whole sustainability of electrosynthetic procedures. Herein, we report …

Herein, we have revealed a methodology for the selective C-alkylation of benzoxazolones,
benzothiazolones, indolinones, and benzimidazolones incorporating activated alcohols …

The benzoxazole is one of the most widely exploited heterocycles in drug discovery. Natural
occurring and synthetic benzoxazoles show a broad range of biological activities. Many …

We herein report the cyclocondensation of o-aminophenols with α-ketothioesters in acidic
media for the highly regioselective synthesis of 2-acylbenzoxazoles in DMF at 80° C. The …

In current study, an efficient and simple synthesis of phenyl-benzoxazoles derivatives (1–14)
were carried out, upon cyclization of 2-aminophenol with substituted aldehyde. All …

The benzoxazole core, featuring a sterically congested 2, 6-disubstituted aryl fragment at the
C2 position, exhibits exclusive three-dimensional structures that are essential for particular …