Current status of N-, O-, S-heterocycles as potential alkaline phosphatase inhibitors: a medicinal chemistry overview

RS Jassas, N Naeem, A Sadiq, R Mehmood… - RSC …, 2023 - pubs.rsc.org
Heterocycles are a class of compounds that have been found to be potent inhibitors of
alkaline phosphatase (AP), an enzyme that plays a critical role in various physiological …

Exploring fluorine-substituted piperidines as potential therapeutics for diabetes mellitus and Alzheimer's diseases

EU Mughal, MB Hawsawi, N Naeem, A Hassan… - European journal of …, 2024 - Elsevier
In the current study, a series of fluorine-substituted piperidine derivatives (1–8) has been
synthesized and characterized by various spectroscopic techniques. In vitro and in vivo …

[HTML][HTML] Synthesis of new bis (dimethylamino) benzophenone hydrazone for diabetic management: In-vitro and in-silico approach

M Khan, G Ahad, A Alam, S Ullah, A Khan, U Salar… - Heliyon, 2024 - cell.com
Inhibiting α-glucosidase is a reliable method for reducing blood sugar levels in diabetic
individuals. Bis (dimethylamino) benzophenone derivatives 1–27 were synthesized from bis …

Novel hydrazones derived from anthranilic acid as potent cholinesterases and α‐glycosidase inhibitors: Synthesis, characterization, and biological effects

FS Tokalı, P Taslimi, T Taskin‐Tok… - … of Biochemical and …, 2024 - Wiley Online Library
N‐substitued anthranilic acid derivatives are commonly found in the structure of many
biologically active molecules. In this study, new members of hydrazones derived from …

Design and synthesis of 2-amino-4,6-diarylpyrimidine derivatives as potent α-glucosidase and α-amylase inhibitors: structure–activity relationship, in vitro, QSAR …

EU Mughal, S Amjid, A Sadiq, N Naeem… - Journal of …, 2024 - Taylor & Francis
In the present study, a series of 2-amino-4, 6-diarylpyrimidine derivatives was designed,
synthesized, characterized and evaluated for their in vitro α-glucosidase and α-amylase …

Synthesis, biological evaluation and molecular modeling studies of modulated benzyloxychalcones as potential acetylcholinesterase inhibitors

A Abdalla Ali, SA Mhamad, AH Hasan… - Journal of …, 2024 - Taylor & Francis
Acetylcholinesterase inhibitors (AChEIs) have become a significant target in the search for
an efficient treatment of Alzheimer's disease. Chalcone-based compounds display a strong …

Synthesis, in vitro α-glucosidase, and acetylcholinesterase inhibitory activities of novel indol-fused pyrano [2, 3-d] pyrimidine compounds

HT Nguyen, AN Tuan, TAD Thi, KT Van… - Bioorganic & Medicinal …, 2024 - Elsevier
In this study, new indol-fused pyrano [2, 3-d] pyrimidines were designed and synthesized.
These products were obtained in moderate to good yields and their structures were …

Synthesis, in vitro β-glucuronidase inhibitory potential and molecular docking study of benzimidazole analogues

H Ullah, A Nawaz, F Rahim, I Uddin, A Hussain… - Chemical Data …, 2023 - Elsevier
We have synthesized fifteen benzimidazole bearing Schiff base analogues (1–15),
characterized through different techniques such as NMR, HR-EIMS and evaluated against β …

Synthesis of zinc phthalocyanine containing 1, 2-phenylene bis (3-chloropropanoate) substituted groups and investigation of their metabolic enzyme inhibitory effects

DG Solğun, N Sadeghian, P Taslimi, T Taskin-Tok… - Polyhedron, 2024 - Elsevier
Abstract In this study, 4, 5-dicyano-1, 2-phenylene dinicotinate compound was obtained as a
result of the reaction of 4, 5-dichlorophthalonitrile and nicotinic acid. This compound was …

Synthesis, in vitro α-glucosidase and α-amylase activities, and an in silico molecular docking study of triazinoindole-thiazolidinone hybrid derivatives

AA Khan, H Ullah, F Rahim, M Taha, F Khan… - Chemical Data …, 2023 - Elsevier
Abstract Triazinoindole-thiazolidinone hybrid derivatives (1–10) was synthesised and
evaluated them against α-glucosidase and α-amylase enzymes. All synthesised derivatives …