Computer-aided drug design and drug discovery: a prospective analysis

SK Niazi, Z Mariam - Pharmaceuticals, 2023 - mdpi.com
In the dynamic landscape of drug discovery, Computer-Aided Drug Design (CADD) emerges
as a transformative force, bridging the realms of biology and technology. This paper …

Automated model building and protein identification in cryo-EM maps

K Jamali, L Käll, R Zhang, A Brown, D Kimanius… - Nature, 2024 - nature.com
Interpreting electron cryo-microscopy (cryo-EM) maps with atomic models requires high
levels of expertise and labour-intensive manual intervention in three-dimensional computer …

Novel artificial intelligence-based approaches for ab initio structure determination and atomic model building for cryo-electron microscopy

MC DiIorio, AW Kulczyk - Micromachines, 2023 - mdpi.com
Single particle cryo-electron microscopy (cryo-EM) has emerged as the prevailing method
for near-atomic structure determination, shedding light on the important molecular …

Steering masked discrete diffusion models via discrete denoising posterior prediction

J Rector-Brooks, M Hasan, Z Peng, Z Quinn… - arxiv preprint arxiv …, 2024 - arxiv.org
Generative modeling of discrete data underlies important applications spanning text-based
agents like ChatGPT to the design of the very building blocks of life in protein sequences …

Evaluating representation learning on the protein structure universe

AR Jamasb, A Morehead, CK Joshi, Z Zhang, K Didi… - Ar**v, 2024 - pmc.ncbi.nlm.nih.gov
We introduce ProteinWorkshop, a comprehensive benchmark suite for representation
learning on protein structures with Geometric Graph Neural Networks. We consider large …

Protein fitness prediction is impacted by the interplay of language models, ensemble learning, and sampling methods

M Mardikoraem, D Woldring - Pharmaceutics, 2023 - mdpi.com
Advances in machine learning (ML) and the availability of protein sequences via high-
throughput sequencing techniques have transformed the ability to design novel diagnostic …

Integrating Embeddings from Multiple Protein Language Models to Improve Protein O-GlcNAc Site Prediction

S Pokharel, P Pratyush, HD Ismail, J Ma… - International Journal of …, 2023 - mdpi.com
O-linked β-N-acetylglucosamine (O-GlcNAc) is a distinct monosaccharide modification of
serine (S) or threonine (T) residues of nucleocytoplasmic and mitochondrial proteins. O …

Fast protein structure searching using structure graph embeddings

JG Greener, K Jamali - bioRxiv, 2022 - biorxiv.org
Comparing and searching protein structures independent of primary sequence has proved
useful for remote homology detection, function annotation and protein classification. With the …

Functional protein dynamics directly from sequences

K Jia, M Kilinc, RL Jernigan - The Journal of Physical Chemistry B, 2023 - ACS Publications
The sequence correlations within a protein multiple sequence alignment are routinely being
used to predict contacts within its structure, but here we point out that these data can also be …

TAFPred: Torsion Angle Fluctuations Prediction from Protein Sequences

MWU Kabir, DM Alawad, A Mishra, MT Hoque - Biology, 2023 - mdpi.com
Simple Summary This study aimed to create an intelligent computer model called TAFPred
to predict how proteins move and twist by looking at their sequences. By analyzing different …