Dearomative dienolate-mediated catalysis: A remote activation strategy for asymmetric functionalization of benzylic C–H bonds of heteroaryl aldehydes
Y Wang, JB Lin, JK **e, H Lu, XQ Hu, PF Xu - Organic letters, 2018 - ACS Publications
A dearomative remote activation strategy for the asymmetric functionalization of benzylic C–
H bonds of heteroaryl aldehydes under bifunctional Brønsted base catalysis has been …
H bonds of heteroaryl aldehydes under bifunctional Brønsted base catalysis has been …
Reduction of interstrand charge repulsion of DNA duplexes by salts and by neutral phosphotriesters–contrary effects for harnessing duplex formation
To exploit the formation of DNA duplexes, the charge repulsion between complementary
DNA strands can be reduced by adding salts or by replacing the negatively charged natural …
DNA strands can be reduced by adding salts or by replacing the negatively charged natural …
Synthesis of Novel pyrimido [4, 5-b] quinoline-4-one Derivatives and Assessment as Antimicrobial and Antioxidant Agents
U Fathy, RS Gouhar, A Younis… - Pharmacognosy …, 2021 - phcogj.com
Objective: Antimicrobial resistance has emerged as one of the serious global health
problems of the 21 st century that threatens the efficient treatment and prevention of an …
problems of the 21 st century that threatens the efficient treatment and prevention of an …
Synthesis and biological evaluation of 4H-benzo [e][1, 3] oxazin-4-ones analogues of TGX-221 as inhibitors of PI3Kβ
EUR Mohammed, ZJ Porter, IG Jennings… - Bioorganic & Medicinal …, 2022 - Elsevier
A novel series of TGX-221 analogues was prepared that include isosteric replacement of the
4H-pyrido [1, 2-a] pyrimidin-4-one with a 4H-benzo [e][1, 3] oxazin-4-one scaffold. The …
4H-pyrido [1, 2-a] pyrimidin-4-one with a 4H-benzo [e][1, 3] oxazin-4-one scaffold. The …
Cycloaddition of 4-Acyl-1H-pyrrole-2,3-diones Fused at [e]-Side and Cyanamides: Divergent Approach to 4H-1,3-Oxazines
EE Khramtsova, AD Krainov, MV Dmitriev… - Molecules, 2022 - mdpi.com
4-Acyl-1 H-pyrrole-2, 3-diones fused at [e]-side with a heterocyclic moiety are suitable
platforms for the development of a hetero-Diels–Alder-reaction-based, diversity-oriented …
platforms for the development of a hetero-Diels–Alder-reaction-based, diversity-oriented …
Novel 6-substituted-2-morpholino-8-(1-(arylamino or aryloxo) ethyl)-4H-benzo [e][1, 3] oxazin-4-ones as Selective PI3K Inhibitors and Anticancer Compounds
E Mohammed - 2021 - opal.latrobe.edu.au
A thesis submitted in total fulfilment of the requirements for the degree of Doctor of
Philosophy to the Department of Pharmacy and Biomedical Sciences, School of Molecular …
Philosophy to the Department of Pharmacy and Biomedical Sciences, School of Molecular …
[CITATION][C] 1, 3-Oxazines and their benzo derivatives
L Lázár, F Fülöp - 2008 - Elsevier