Review on potential biological activities of thiosemicarbazides

S Singhal, S Arora, S Agarwal, R Sharma, N Singhal - 2013 - dr.ddn.upes.ac.in
Heterocycles have contributed to the development of society from a biological and industrial
point of view as well as to improve the quality of life. During the past few decades, interest …

Transalkylidation reaction: Green, catalyst-free synthesis of thiosemicarbazones and solving the NMR conflict between their acyclic structure and intramolecular …

MA El-Atawy, AZ Omar, M Hagar… - Green Chemistry Letters …, 2019 - Taylor & Francis
ABSTRACT A series of arylidene thiosemicarbazides have been prepared by a new method,
which was titled as transalkylidation. This method is an effective, fast, green and clean …

Exploring molecular structure, spectral features, electronic properties and molecular docking of a novel biologically active heterocyclic compound 4 …

R Arivazhagan, C Sridevi, A Prakasam - Journal of Molecular Structure, 2021 - Elsevier
The experimental and theoretical studies on the structure and vibrations of 4-phenyl
thiosemicarbazide (PTSC)(IUPAC: 3-amino-1-phenylthiourea) have been carried out using …

[HTML][HTML] Synthesis and anthelmintic activity of new thiosemicarbazide derivatives—A preliminary study

K Dziduch, P Kołodziej, A Paneth, A Bogucka-Kocka… - Molecules, 2020 - mdpi.com
Parasitic infections caused by different species of intestinal helminths still poses a threat to
public health. There is a need to search for new, effective anthelmintic drugs. A series of …

Studies on isoniazid derivatives through a medicinal chemistry approach for the identification of new inhibitors of urease and inflammatory markers

F Rizvi, M Khan, A Jabeen, H Siddiqui… - Scientific Reports, 2019 - nature.com
A library of thiosemicarbazide derivatives of isoniazid 3–27, was synthesized and evaluated
for their anti-inflammatory and urease inhibition activities, by using in vitro bioassays. Among …

Novel thiosemicarbazide–oxadiazole hybrids as unprecedented inhibitors of yeast α-glucosidase and in silico binding analysis

M Taha, NH Ismail, S Imran, A Wadood, M Ali… - RSC Advances, 2016 - pubs.rsc.org
Compounds 1–18, new oxadiazole–thiosemicarbazide hybrids, were synthesized using a
five-step reaction sequence in excellent yields. All the synthesized analogs exhibited …

[HTML][HTML] Supramolecular aggregation of lead (II) perchlorate and a thiosemicarbazide derivative linked by a myriad of non-covalent interactions

I García-Santos, A Castineiras, G Mahmoudi… - Inorganica Chimica …, 2022 - Elsevier
In this work, we report on a new lead (II) coordination complex [Pb 2 L 2 (CH 3 CN)(ClO 4)
2]· 2H 2 O (1· 2H 2 O), which was readily synthesized from a mixture of Pb (ClO 4) 2· 3H 2 O …

Ultrasonic-assisted synthesis of amantadine derivatives-in vitro urease and α-glucosidase inhibitory activities, mechanistic, and computational studies

M Raza, H Siddiqui, M Khan, S Ullah, F Rizvi… - Journal of Molecular …, 2022 - Elsevier
Ultrasonic synthesis of 26 amantadine derivatives,(3-28) including seven new compounds,
are reported with significantly reduced synthesis time and increased percentage yield …

Rationally designed hecogenin thiosemicarbazone analogs as novel MEK inhibitors for the control of breast malignancies

HE Elsayed, HY Ebrahim, EG Haggag… - Bioorganic & Medicinal …, 2017 - Elsevier
Natural products have documented oncology success history as valuable scaffolds for
selective target modulation. Herein, the sapogenin hecogenin (1) was screened for its anti …

New Thiosemicarbazide Derivatives with Multidirectional Biological Action

P Lasek, U Kosikowska, P Kołodziej… - Molecules, 2024 - mdpi.com
Over the years, several new medicinal substances have been introduced for the treatment of
diseases caused by bacteria and parasites. Unfortunately, due to the production of …