[HTML][HTML] Molecular and clinical aspects of potential neurotoxicity induced by new psychoactive stimulants and psychedelics

D Rudin, ME Liechti, D Luethi - Experimental neurology, 2021‏ - Elsevier
New psychoactive stimulants and psychedelics continue to play an important role on the
illicit new psychoactive substance (NPS) market. Designer stimulants and psychedelics both …

Reinstatement of synaptic plasticity in the aging brain through specific dopamine transporter inhibition

J Lubec, P Kalaba, AM Hussein, DD Feyissa, MH Kotob… - 2021‏ - nature.com
Aging-related neurological deficits negatively impact mental health, productivity, and social
interactions leading to a pronounced socioeconomic burden. Since declining brain …

The interaction of organic cation transporters 1-3 and PMAT with psychoactive substances

J Maier, M Niello, D Rudin, LC Daws… - Organic cation transporters …, 2021‏ - Springer
Abstract Organic cation transporters 1-3 (OCT1-3, SLC22A1-3) and the plasma membrane
monoamine transporter (PMAT, SLC29A4) play a major role in maintaining monoaminergic …

Differentiated HT22 cells as a novel model for in vitro screening of serotonin reuptake inhibitors

J Lim, Y Bang, KM Kim, HJ Choi - Frontiers in Pharmacology, 2023‏ - frontiersin.org
The mouse hippocampal neuronal cell line HT22 is frequently used as an in vitro model to
investigate the role of hippocampal cholinergic neurons in cognitive functions. HT22 cells …

[HTML][HTML] α-PPP and its derivatives are selective partial releasers at the human norepinephrine transporter: a pharmacological characterization of interactions between …

J Maier, L Rauter, D Rudin, M Niello, M Holy… - …, 2021‏ - Elsevier
While classical cathinones, such as methcathinone, have been shown to be monoamine
releasing agents at human monoamine transporters, the subgroup of α-pyrrolidinophenones …

Pharmacological characterization of toludesvenlafaxine as a triple reuptake inhibitor

H Zhu, W Wang, C Sha, W Guo, C Li, F Zhao… - Frontiers in …, 2021‏ - frontiersin.org
Toludesvenlafaxine hydrochloride dihydrate is a novel chemical entity and a potential triple
monoamine reuptake inhibitor. This study characterized the in vitro triple reuptake inhibition …

Bioisosteric analogs of MDMA: Improving the pharmacological profile?

AS Alberto‐Silva, S Hemmer, HA Bock… - Journal of …, 2024‏ - Wiley Online Library
Methylenedioxymethamphetamine (MDMA,'ecstasy') is re‐emerging in clinical settings as a
candidate for the treatment of specific neuropsychiatric disorders (eg post‐traumatic stress …

Characterization of neurotransmitter inhibition for seven cathinones by a proprietary fluorescent dye method

M Persson, S Vikingsson, R Kronstrand… - Drug Testing and …, 2024‏ - Wiley Online Library
Many new psychoactive substances (NPS) are stimulants, and information about their
potency and abuse potential is often lacking. To start addressing this need, a method …

Interaction profiles of central nervous system active drugs at human organic cation transporters 1–3 and human plasma membrane monoamine transporter

TJF Angenoorth, S Stankovic, M Niello, M Holy… - International Journal of …, 2021‏ - mdpi.com
Many psychoactive compounds have been shown to primarily interact with high-affinity and
low-capacity solute carrier 6 (SLC6) monoamine transporters for norepinephrine (NET; …

Effects of Hydroxylated Mephedrone Metabolites on Monoamine Transporter Activity in vitro

M Niello, D Cintulová, P Raithmayr, M Holy… - Frontiers in …, 2021‏ - frontiersin.org
Mephedrone is a largely abused psychostimulant. It elicits the release of monoamines via
the high affinity transporters for dopamine (DAT), norepinephrine (NET) and serotonin …