[HTML][HTML] Pharmaceutical amorphous solid dispersion: A review of manufacturing strategies

SV Bhujbal, B Mitra, U Jain, Y Gong, A Agrawal… - … Pharmaceutica Sinica B, 2021 - Elsevier
Amorphous solid dispersions (ASDs) are popular for enhancing the solubility and
bioavailability of poorly water-soluble drugs. Various approaches have been employed to …

Amorphous solid dispersions: Rational selection of a manufacturing process

T Vasconcelos, S Marques, J das Neves… - Advanced drug delivery …, 2016 - Elsevier
Amorphous products and particularly amorphous solid dispersions are currently one of the
most exciting areas in the pharmaceutical field. This approach presents huge potential and …

Current trends and future perspectives of solid dispersions containing poorly water-soluble drugs

CLN Vo, C Park, BJ Lee - European journal of pharmaceutics and …, 2013 - Elsevier
Over 40% of active pharmaceutical ingredients (API) in development pipelines are poorly
water-soluble drugs which limit formulation approaches, clinical application and …

Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs

T Vasconcelos, B Sarmento, P Costa - Drug discovery today, 2007 - Elsevier
Solid dispersions are one of the most promising strategies to improve the oral bioavailability
of poorly water soluble drugs. By reducing drug particle size to the absolute minimum, and …

Eutectic mixtures as an approach to enhance solubility, dissolution rate and oral bioavailability of poorly water-soluble drugs

GC Bazzo, BR Pezzini, HK Stulzer - International Journal of Pharmaceutics, 2020 - Elsevier
Eutectic mixtures have been known for a long time in the pharmaceutical field. However, its
potential as a system to improve the solubility and dissolution of poorly water-soluble drugs …

Preparation and evaluation of nanosuspensions for enhancing the dissolution of poorly soluble drugs

P Kocbek, S Baumgartner, J Kristl - International journal of pharmaceutics, 2006 - Elsevier
Poorly water-soluble compounds are difficult to develop as drug products using
conventional formulation techniques and are frequently abandoned early in discovery. In the …

The preparation of orally disintegrating tablets using a hydrophilic waxy binder

G Abdelbary, P Prinderre, C Eouani, J Joachim… - International journal of …, 2004 - Elsevier
The demand for rapidly disintegrating tablets (RDT) has been growing during the last
decade especially for elderly and children who have swallowing difficulties. The problem of …

Preparation, characterization and in vivo evaluation of ibuprofen binary solid dispersions with poloxamer 188

M Newa, KH Bhandari, DX Li, TH Kwon, JA Kim… - International journal of …, 2007 - Elsevier
Ibuprofen–Poloxamer 188 (P 188) binary solid dispersions (SD) with different drug loadings
were prepared, characterized by scanning electron microscopy (SEM), differential scanning …

[HTML][HTML] Classification of scanning electron microscope images of pharmaceutical excipients using deep convolutional neural networks with transfer learning

H Iwata, Y Hayashi, A Hasegawa, K Terayama… - International Journal of …, 2022 - Elsevier
Abstract Convolutional Neural Networks (CNNs) are image analysis techniques that have
been applied to image classification in various fields. In this study, we applied a CNN to …

Evaluation of melt granulation and ultrasonic spray congealing as techniques to enhance the dissolution of praziquantel

N Passerini, B Albertini, B Perissutti… - International journal of …, 2006 - Elsevier
Praziquantel (PZQ), an anthelminthic drug widely used in develo** countries, is classified
in Class II in the Biopharmaceutics Classification Systems; this means that PZQ has very low …