Conspectus Late-stage halogenation, targeting specific positions in complex substrates, has
gained significant attention due to its potential for diversifying and functionalizing complex …

Conspectus The selective functionalization/transformation of ubiquitous pyridine-fused N-
heteroarenes is a practical method to synthesize structurally novel N-heterocycles, which is …

Aromatic electron-deficient heterocycles, such as pyridines, are found in many biologically
relevant structures, including those with medicinal applications. Methods for their …

A highly effective external photocatalyst-and additive-free method for the phosphorylation of
3, 4-dihydroquinoxalin-2 (1 H)-ones to produce phosphorylated dihydroquinoxalin-2 (1 H) …

Considering the indispensable significance and utilities of meta-substituted pyridines in
medicinal, chemical as well as materials science, a direct meta-selective C–H …

Herein, we report a one‐pot method for enantioselective C− H allylation of pyridines at C3
via tandem borane and palladium catalysis. This method involves borane‐catalyzed …

In this report, we developed a unified and standardized one-pot sequence that converts
pyridine derivatives into 1, 2-diazepines by inserting a nitrogen atom. This skeletal …

Direct C–H fluorination is an efficient strategy to construct aromatic C–F bonds, but the
cleavage of specific C–H bonds in the presence of other functional groups and the high …

The C–H hydroxylation of the pyridine C3 position is a highly desirable transformation but
remains a great challenge due to the inherent electronic properties of this heterocycle core …

Methods to incorporate stable radioisotopes are integral to pharmaceutical and
agrochemical development. However, despite the prevalence of pyridines in candidate …