[HTML][HTML] Glucagon-like peptide 1 (GLP-1)

TD Müller, B Finan, SR Bloom, D D'Alessio… - Molecular …, 2019‏ - Elsevier
Background The glucagon-like peptide-1 (GLP-1) is a multifaceted hormone with broad
pharmacological potential. Among the numerous metabolic effects of GLP-1 are the glucose …

The discovery and development of liraglutide and semaglutide

LB Knudsen, J Lau - Frontiers in endocrinology, 2019‏ - frontiersin.org
The discovery of glucagon-like peptide-1 (GLP-1), an incretin hormone with important effects
on glycemic control and body weight regulation, led to efforts to extend its half-life and make …

Discovery of the once-weekly glucagon-like peptide-1 (GLP-1) analogue semaglutide

J Lau, P Bloch, L Schäffer, I Pettersson… - Journal of medicinal …, 2015‏ - ACS Publications
Liraglutide is an acylated glucagon-like peptide-1 (GLP-1) analogue that binds to serum
albumin in vivo and is approved for once-daily treatment of diabetes as well as obesity. The …

Effects of once‐weekly semaglutide on appetite, energy intake, control of eating, food preference and body weight in subjects with obesity

J Blundell, G Finlayson, M Axelsen… - Diabetes, Obesity …, 2017‏ - Wiley Online Library
Aim The aim of this trial was to investigate the mechanism of action for body weight loss with
semaglutide. Materials and methods This randomised, double‐blind, placebo‐controlled …

The impact of short-chain fatty acids on GLP-1 and PYY secretion from the isolated perfused rat colon

CB Christiansen, MBN Gabe… - American Journal …, 2018‏ - journals.physiology.org
The colonic epithelium harbors a large number of endocrine cells, but little is known about
the endocrine functions of the colon. However, the high density of glucagon like peptide-1 …

Incretin drugs in diabetic kidney disease: biological mechanisms and clinical evidence

RZ Alicic, EJ Cox, JJ Neumiller, KR Tuttle - Nature Reviews Nephrology, 2021‏ - nature.com
As the prevalence of diabetes continues to climb, the number of individuals living with
diabetic complications will reach an unprecedented magnitude. The emergence of new …

Pharmacology and therapeutic implications of current drugs for type 2 diabetes mellitus

AA Tahrani, AH Barnett, CJ Bailey - Nature Reviews Endocrinology, 2016‏ - nature.com
Type 2 diabetes mellitus (T2DM) is a global epidemic that poses a major challenge to health-
care systems. Improving metabolic control to approach normal glycaemia (where practical) …

Severe obesity in children and adolescents: identification, associated health risks, and treatment approaches: a scientific statement from the American Heart …

AS Kelly, SE Barlow, G Rao, TH Inge, LL Hayman… - Circulation, 2013‏ - Am Heart Assoc
Severe obesity afflicts between 4% and 6% of all youth in the United States, and the
prevalence is increasing. Despite the serious immediate and long-term cardiovascular …

GLP-1 receptor agonists for individualized treatment of type 2 diabetes mellitus

JJ Meier - Nature Reviews Endocrinology, 2012‏ - nature.com
In healthy humans, the incretin glucagon-like peptide 1 (GLP-1) is secreted after eating and
lowers glucose concentrations by augmenting insulin secretion and suppressing glucagon …

[HTML][HTML] Exenatide once weekly for alcohol use disorder investigated in a randomized, placebo-controlled clinical trial

MK Klausen, ME Jensen, M Møller, N Le Dous… - JCI insight, 2022‏ - ncbi.nlm.nih.gov
Background Alcohol use disorder (AUD) is a chronic, relapsing brain disorder that accounts
for 5% of deaths annually, and there is an urgent need to develop new targets for …