The effect of cyclophosphamide on the immune system: implications for clinical cancer therapy

M Ahlmann, G Hempel - Cancer chemotherapy and pharmacology, 2016 - Springer
Cyclophosphamide is an alkylating agent belonging to the group of oxazaphosporines. As
cyclophosphamide is in clinical use for more than 40 years, there is a lot of experience using …

ABC transporter-mediated multidrug-resistant cancer

H Amawi, HM Sim, AK Tiwari, SV Ambudkar… - Drug transporters in …, 2019 - Springer
ATP-binding cassette (ABC) transporters are involved in active pum** of many diverse
substrates through the cellular membrane. The transport mediated by these proteins …

Anti-SARS-CoV-2 Activity of Andrographis paniculata Extract and Its Major Component Andrographolide in Human Lung Epithelial Cells and Cytotoxicity Evaluation …

K Sa-Ngiamsuntorn, A Suksatu… - Journal of natural …, 2021 - ACS Publications
The coronaviruses disease 2019 (COVID-19) caused by a novel coronavirus (SARS-CoV-2)
has become a major health problem, affecting more than 50 million people with over one …

SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules

A Daina, O Michielin, V Zoete - Scientific reports, 2017 - nature.com
To be effective as a drug, a potent molecule must reach its target in the body in sufficient
concentration, and stay there in a bioactive form long enough for the expected biologic …

Medicinal chemistry strategies to discover P-glycoprotein inhibitors: An update

J Dong, Z Qin, WD Zhang, G Cheng, AG Yehuda… - Drug Resistance …, 2020 - Elsevier
The presence of multidrug resistance (MDR) in malignant tumors is one of the primary
causes of treatment failure in cancer chemotherapy. The overexpression of the ATP binding …

A novel chemometric method for the prediction of human oral bioavailability

X Xu, W Zhang, C Huang, Y Li, H Yu, Y Wang… - International journal of …, 2012 - mdpi.com
Orally administered drugs must overcome several barriers before reaching their target site.
Such barriers depend largely upon specific membrane transport systems and intracellular …

ATP‐binding cassette (ABC) transporters in cancer: A review of recent updates

JQ Wang, ZX Wu, Y Yang, QX Teng… - Journal of Evidence …, 2021 - Wiley Online Library
The ATP‐binding cassette (ABC) transporter superfamily is one of the largest membrane
protein families existing in wide spectrum of organisms from prokaryotes to human. ABC …

Emergence and spread of antibiotic-resistant foodborne pathogens from farm to table

J Kim, J Ahn - Food Science and Biotechnology, 2022 - Springer
Antibiotics have been overused and misused for preventive and therapeutic purposes.
Specifically, antibiotics are frequently used as growth promoters for improving productivity …

Computational analysis of calculated physicochemical and ADMET properties of protein-protein interaction inhibitors

D Lagorce, D Douguet, MA Miteva, BO Villoutreix - Scientific reports, 2017 - nature.com
The modulation of PPIs by low molecular weight chemical compounds, particularly by orally
bioavailable molecules, would be very valuable in numerous disease indications. However …

An overview of the evidence and mechanisms of herb–drug interactions

PS Fasinu, PJ Bouic, B Rosenkranz - Frontiers in pharmacology, 2012 - frontiersin.org
Despite the lack of sufficient information on the safety of herbal products, their use as
alternative and/or complementary medicine is globally popular. There is also an increasing …