Update on the pharmacology of calcitonin/CGRP family of peptides: IUPHAR Review 25

DL Hay, ML Garelja, DR Poyner… - British journal of …, 2018 - Wiley Online Library
The calcitonin/CGRP family of peptides includes calcitonin, α and β CGRP, amylin,
adrenomedullin (AM) and adrenomedullin 2/intermedin (AM2/IMD). Their receptors consist …

Vascular actions of calcitonin gene-related peptide and adrenomedullin

SD Brain, AD Grant - Physiological reviews, 2004 - journals.physiology.org
This review summarizes the receptor-mediated vascular activities of calcitonin gene-related
peptide (CGRP) and the structurally related peptide adrenomedullin (AM). CGRP is a 37 …

A structural basis for amylin receptor phenotype

J Cao, MJ Belousoff, YL Liang, RM Johnson… - Science, 2022 - science.org
Amylin receptors (AMYRs) are heterodimers of the calcitonin (CT) receptor (CTR) and one of
three receptor activity–modifying proteins (RAMPs), AMY1R, AMY2R, and AMY3R. Selective …

Neuropeptides, food intake and body weight regulation: a hypothalamic focus

JJG Hillebrand, D De Wied, RAH Adan - Peptides, 2002 - Elsevier
Energy homeostasis is controlled by a complex neuroendocrine system consisting of
peripheral signals like leptin and central signals, in particular, neuropeptides. Several …

The anorectic effect of a chronic peripheral infusion of amylin is abolished in area postrema/nucleus of the solitary tract (AP/NTS) lesioned rats

TA Lutz, A Mollet, PA Rushing, T Riediger… - International journal of …, 2001 - nature.com
OBJECTIVE: Neurons in the area postrema/nucleus of the solitary tract (AP/NTS) region
mediate amylin's anorectic effect elicited by a single intraperitoneal (ip) injection of a low …

Mediators of amylin action in metabolic control

CN Boyle, Y Zheng, TA Lutz - Journal of clinical medicine, 2022 - mdpi.com
Amylin (also called islet amyloid polypeptide (IAPP)) is a pancreatic beta-cell hormone that
is co-secreted with insulin in response to nutrient stimuli. The last 35 years of intensive …

[HTML][HTML] Gut-brain axis and addictive disorders: A review with focus on alcohol and drugs of abuse

E Jerlhag - Pharmacology & Therapeutics, 2019 - Elsevier
Due to the limited efficacy of existing medications for addictive disorders including alcohol
use disorder (AUD), the need for additional medications is substantial. Potential new …

Control of energy homeostasis by amylin

TA Lutz - Cellular and molecular life sciences, 2012 - Springer
Amylin is an important control of nutrient fluxes because it reduces energy intake, modulates
nutrient utilization by inhibiting postprandial glucagon secretion, and increases energy …

Amylin and calcitonin: potential therapeutic strategies to reduce body weight and liver fat

DS Mathiesen, A Lund, T Vilsbøll, FK Knop… - Frontiers in …, 2021 - frontiersin.org
The hormones amylin and calcitonin interact with receptors within the same family to exert
their effects on the human organism. Calcitonin, derived from thyroid C cells, is known for its …

Infusion of the amylin antagonist AC 187 into the area postrema increases food intake in rats

A Mollet, S Gilg, T Riediger, TA Lutz - Physiology & behavior, 2004 - Elsevier
According to previous studies, the area postrema (AP) of the hindbrain may play an
important role in mediating the anorectic effect of the pancreatic hormone amylin. Peripheral …