Recent advancement of piperidine moiety in treatment of cancer-A review

P Goel, O Alam, MJ Naim, F Nawaz, M Iqbal… - European journal of …, 2018‏ - Elsevier
Piperidine is an important pharmacophore, a privileged scaffold and an excellent
heterocyclic system in the field of drug discovery which provides numerous opportunities in …

Alkaloids from apocynaceae: origin, pharmacotherapeutic properties, and structure-activity studies

A Dey, A Mukherjee, M Chaudhury - Studies in natural products chemistry, 2017‏ - Elsevier
Alkaloids are a diverse group of naturally occurring secondary compounds derived from
amino acids or the process of transamination. Some synthetic compounds with similar …

Palladium‐catalyzed regioselective aromatic extension of internal alkynes through a norbornene‐controlled reaction sequence

Q Zhao, WC Fu, FY Kwong - Angewandte Chemie, 2018‏ - Wiley Online Library
A regioselective aromatic π‐extension reaction of internal alkynes is reported. The proposed
method employs three easily available components, namely aryl halides, 2 …

Iodide-Dependent Selective Dehydroaromatization Affording Maleimide-Fused 9, 10-Phenanthrenes and Their Analogues

S Wang, Z Chen, S Chen, W Shao, Y Chen… - Organic …, 2023‏ - ACS Publications
A novel and selective synthesis of polycyclic fused maleimides from easily available raw
materials under metal-free conditions is presented. This cascade protocol involves self …

Design, synthesis, and biological activity of sulfonamide analogues of antofine and cryptopleurine as potent and orally active antitumor agents

Y Kwon, J Song, H Lee, EY Kim, K Lee… - Journal of Medicinal …, 2015‏ - ACS Publications
Due to their profound antiproliferative activity and unique mode of action,
phenanthroindolizidine and phenanthroquinolizidine alkaloids, represented by antofine and …

Pd-Catalyzed Alkene-Relayed Intermolecular C–H Alkylation Using Aryl Halide Substrates

S Yang, Y Zhang - Organic Letters, 2022‏ - ACS Publications
Alkene-relayed C–H activation represents a novel strategy for functionalizing C–H bonds
selectively. We developed a Pd-catalyzed annulation reaction of 2-iodobiphenyls with …

Design, synthesis, and antiviral evaluation of phenanthrene-based tylophorine derivatives as potential antiviral agents

K Wang, Y Hu, Y Liu, N Mi, Z Fan, Y Liu… - Journal of agricultural …, 2010‏ - ACS Publications
A series of C9-substituted phenanthrene-based tylophorine derivatives (PBTs) were
designed, synthesized, and first evaluated for their antiviral activities against tobacco mosaic …

Multi-omics strategy reveals that Cordyceps sinensis ameliorates sepsis-associated acute kidney injury via reprogramming of mitochondrial energy metabolism and …

L Chen, T Yang, J Wu, G Cheng, M Zhao… - Acta Materia …, 2024‏ - scienceopen.com
Cordyceps sinensis (CS) has been widely used as a dietary supplement or traditional
medicine for the prevention, treatment, and prognostication of various diseases, because of …

Alkaloids as anticancer agents: a review of Chinese patents in recent 5 years

H Tao, L Zuo, H Xu, C Li, G Qiao… - Recent Patents on Anti …, 2020‏ - benthamdirect.com
Background: In recent years, many novel alkaloids with anticancer activity have been found
in China, and some of them are promising for develo** as anticancer agents. Objective …

Directed Metalation–Suzuki–Miyaura Cross-Coupling Strategies: Regioselective Synthesis of Hydroxylated 1-Methyl-phenanthrenes

KB Jørgensen, T Rantanen, T Dörfler… - The Journal of Organic …, 2015‏ - ACS Publications
A general, efficient, and regioselective synthesis of a series of hydroxylated 1-
methylphenanthrenes 9 by a combined directed ortho metalation (DoM)–Suzuki–Miyaura …