New insights into activation and function of the AMPK

GR Steinberg, DG Hardie - Nature reviews Molecular cell biology, 2023 - nature.com
The classical role of AMP-activated protein kinase (AMPK) is as a cellular energy sensor
activated by falling energy status, signalled by increases in AMP to ATP and ADP to ATP …

AMP-activated protein kinase: the current landscape for drug development

GR Steinberg, D Carling - Nature reviews Drug discovery, 2019 - nature.com
Since the discovery of AMP-activated protein kinase (AMPK) as a central regulator of energy
homeostasis, many exciting insights into its structure, regulation and physiological roles …

AMPK: an energy-sensing pathway with multiple inputs and outputs

DG Hardie, BE Schaffer, A Brunet - Trends in cell biology, 2016 - cell.com
AMP-activated protein kinase (AMPK) is a key regulator of energy balance expressed
ubiquitously in eukaryotic cells. Here we review the canonical adenine nucleotide …

AMPK as a therapeutic target for treating metabolic diseases

EA Day, RJ Ford, GR Steinberg - Trends in Endocrinology & Metabolism, 2017 - cell.com
The AMP-activated protein kinase (AMPK) is a central regulator of multiple metabolic
pathways and may have therapeutic importance for treating obesity, insulin resistance, type …

Single phosphorylation sites in Acc1 and Acc2 regulate lipid homeostasis and the insulin-sensitizing effects of metformin

MD Fullerton, S Galic, K Marcinko, S Sikkema… - Nature medicine, 2013 - nature.com
The obesity epidemic has led to an increased incidence of nonalcoholic fatty liver disease
(NAFLD) and type 2 diabetes. AMP-activated protein kinase (Ampk) regulates energy …

AMPK and the adaptation to exercise

HR Spaulding, Z Yan - Annual review of physiology, 2022 - annualreviews.org
Noncommunicable diseases are chronic diseases that contribute to death worldwide, but
these diseases can be prevented and mitigated with regular exercise. Exercise activates …

[HTML][HTML] AMPK in skeletal muscle function and metabolism

R Kjøbsted, JR Hingst, J Fentz, M Foretz… - The FASEB …, 2018 - ncbi.nlm.nih.gov
Skeletal muscle possesses a remarkable ability to adapt to various physiologic conditions.
AMPK is a sensor of intracellular energy status that maintains energy stores by fine-tuning …

AMPK activators: mechanisms of action and physiological activities

J Kim, G Yang, Y Kim, J Kim, J Ha - Experimental & molecular medicine, 2016 - nature.com
AMP-activated protein kinase (AMPK) is a central regulator of energy homeostasis, which
coordinates metabolic pathways and thus balances nutrient supply with energy demand …

Inhibiting peripheral serotonin synthesis reduces obesity and metabolic dysfunction by promoting brown adipose tissue thermogenesis

JD Crane, R Palanivel, EP Mottillo, AL Bujak, H Wang… - Nature medicine, 2015 - nature.com
Abstract Mitochondrial uncoupling protein 1 (UCP1) is enriched within interscapular brown
adipose tissue (iBAT) and beige (also known as brite) adipose tissue,, but its thermogenic …

[HTML][HTML] Sarcopenia and muscle aging: a brief overview

T Dao, AE Green, YA Kim, SJ Bae… - Endocrinology and …, 2020 - synapse.koreamed.org
The world is facing the new challenges of an aging population, and understanding the
process of aging has therefore become one of the most important global concerns …