Palladium-catalysed oxidation of primary and secondary alcohols

J Muzart - Tetrahedron, 2003 - Elsevier
The transformation of the hydroxy group into the corresponding carbonyl is one of the most
frequently used reactions in organic synthesis. Traditionally, stoichiometric and even over …

Bicyclic conformationally restricted diamines

OO Grygorenko, DS Radchenko… - Chemical …, 2011 - ACS Publications
The term “conformational restriction” can be found very often in contemporary chemical
literature. Despite the lack of strict definitions, this term is usually intuitively understood and …

Chemoselective reductive aminations in aqueous nanoreactors using parts per million level Pd/C catalysis

RR Thakore, BS Takale, G Casotti, ES Gao… - Organic …, 2020 - ACS Publications
Condensation in recyclable water between aldehydes or ketones and amines occurs
smoothly within the hydrophobic cores of nanomicelles, resulting in imine formation that is …

One-Pot Reductive Mono-N-alkylation of Aniline and Nitroarene Derivatives Using Aldehydes

E Byun, B Hong, KA De Castro, M Lim… - The Journal of organic …, 2007 - ACS Publications
One-pot reductive mono-N-alkylation of aniline and nitroarene derivatives using various
aldehydes by Pd/C catalyst in aqueous 2-propanol solvent with ammonium formate as in situ …

Two-step synthesis of achiral dispiro-1, 2, 4, 5-tetraoxanes with outstanding antimalarial activity, low toxicity, and high-stability profiles

GL Ellis, R Amewu, S Sabbani, PA Stocks… - Journal of medicinal …, 2008 - ACS Publications
A rapid, two-step synthesis of a range of dispiro-1, 2, 4, 5-tetraoxanes with potent
antimalarial activity both in vitro and in vivo has been achieved. These 1, 2, 4, 5-tetraoxanes …

Monanchocidins B–E: Polycyclic Guanidine Alkaloids with Potent Antileukemic Activities from the Sponge Monanchora pulchra

TN Makarieva, KM Tabakmaher, AG Guzii… - Journal of Natural …, 2011 - ACS Publications
New unusual polycyclic guanidine alkaloids monanchocidins B–E (2–5) along with
monanchocidin A (1), which we recently described, were isolated from the Far-Eastern …

Domino hydrogenation–reductive amination of phenols, a simple process to access substituted cyclohexylamines

VR Jumde, E Petricci, C Petrucci, N Santillo… - Organic …, 2015 - ACS Publications
Phenols can be efficiently reduced by sodium formate and Pd/C as the catalyst in water and
in the presence of amines to give the corresponding cyclohexylamines. This reaction works …

Facile preparation of tetrahydro-5H-pyrido [1, 2, 3-de]-1, 4-benzoxazines via reductive cyclization of 2-(8-quinolinyloxy) ethanones and their antioxidant activity

VP Patil, VL Markad, KM Kodam… - Bioorganic & medicinal …, 2013 - Elsevier
Facile preparation of tetrahydro-5H-pyrido[1,2,3-de]-1,4-benzoxazines via reductive
cyclization of 2-(8-quinolinyloxy)ethanones and their antioxidant activity - ScienceDirect …

Direct, Two-Step Synthetic Pathway to Novel Dibenzo[a,c]phenanthridines

F Churruca, R SanMartin, M Carril… - The Journal of …, 2005 - ACS Publications
Novel dibenzo [a, c] phenanthridines are prepared regioselectively by the application of a
straightforward synthetic pathway, starting from new 3, 4-diaryl-and 3, 4-dihydro-3, 4 …

Design and synthesis of diazatricyclodecane agonists of the G-protein-coupled receptor 119

E Darout, RP Robinson, KF McClure… - Journal of Medicinal …, 2013 - ACS Publications
A series of GPR119 agonists based on a 2, 6-diazatricyclo [3.3. 1.1∼ 3, 7∼] decane ring
system is described. Also provided is a detailed account of the development of a multigram …