Thiophene-based derivatives as anticancer agents: An overview on decade's work

S Pathania, PA Chawla - Bioorganic Chemistry, 2020‏ - Elsevier
Heterocyclic compounds hold a pivotal place in medicinal chemistry due to their wide range
of biological activities and thus, are exhaustively explored in the field of drug design and …

Therapeutic potential of oxadiazole or furadiazole containing compounds

A Siwach, PK Verma - BMC chemistry, 2020‏ - Springer
As we know that, Oxadiazole or furadi azole ring containing derivatives are an important
class of heterocyclic compounds. A heterocyclic five-membered ring that possesses two …

Synthesis, biological evaluation, and molecular docking of novel azolylhydrazonothiazoles as potential anticancer agents

JY Al-Humaidi, SM Gomha, SM Riyadh, MS Ibrahim… - ACS …, 2023‏ - ACS Publications
A novel set of thiazolylhydrazonothiazoles bearing an indole moiety were synthesized by
subjection reactions of carbothioamide derivative and hydrazonoyl chlorides (or α …

Pyrimidine: An elite heterocyclic leitmotif in drug discovery‐synthesis and biological activity

S Nadar, T Khan - Chemical Biology & Drug Design, 2022‏ - Wiley Online Library
Heterocyclic compounds bearing the pyrimidine core are of tremendous interest as they
constitute an important class of natural and synthetic compounds exhibiting diverse useful …

Determination of potential inhibitors based on isatin derivatives against SARS-CoV-2 main protease (mpro): a molecular docking, molecular dynamics and structure …

VN Badavath, A Kumar, PK Samanta… - Journal of …, 2022‏ - Taylor & Francis
Abstract SARS-COV-2, the novel coronavirus and root of global pandemic COVID-19
caused a severe health threat throughout the world. Lack of specific treatments raised an …

Synthesis, antiproliferative and apoptosis induction potential activities of novel bis (indolyl) hydrazide-hydrazone derivatives

R Sreenivasulu, KT Reddy, P Sujitha, CG Kumar… - Bioorganic & medicinal …, 2019‏ - Elsevier
In recent years, indole-indazolyl hydrazide-hydrazone derivatives with strong cell growth
inhibition and apoptosis induction characteristics are being strongly screened for their …

[HTML][HTML] Synthesis, molecular docking study, and cytotoxic activity against MCF cells of new Thiazole–Thiophene scaffolds

SM Gomha, SM Riyadh, B Huwaimel, MEM Zayed… - Molecules, 2022‏ - mdpi.com
Investigating novel compounds that may be useful in designing new, less toxic, selective,
and potent breast anticancer agents is still the main challenge for medicinal chemists. Thus …

Design, synthesis, and biological evaluation of chalcone-linked thiazole-imidazopyridine derivatives as anticancer agents

VR Suma, R Sreenivasulu, MVB Rao… - Medicinal Chemistry …, 2020‏ - Springer
A novel library of chalcone linked thiazole-imidazopyridine (12a–j) derivatives were
designed, synthesized, and their structures were characterized by 1 H NMR, 13 C NMR and …

Design, synthesis, and biological evaluation of 1, 2, 4-thiadiazole-1, 2, 4-triazole derivatives bearing amide functionality as anticancer agents

YJ Pragathi, R Sreenivasulu, D Veronica… - Arabian journal for …, 2021‏ - Springer
A novel library of amide functionality having 1, 2, 4-thiadiazole-1, 2, 4-triazole (8a–j) analogs
was designed, synthesized, and structures were characterized by 1 H NMR, 13 C NMR, and …

Synthesis, anticancer evaluation and molecular docking studies of 2, 5-bis (indolyl)-1, 3, 4-oxadiazoles, Nortopsentin analogues

R Sreenivasulu, MB Tej, SS Jadav, P Sujitha… - Journal of Molecular …, 2020‏ - Elsevier
A series of ten novel 2, 5-bis (indolyl)-1, 3, 4-oxadiazoles were designed and synthesized.
All these compounds were evaluated for their cytotoxicity against four cancer cell lines …