Targeting Tau hyperphosphorylation via kinase inhibition: strategy to address Alzheimer's disease

AA Turab Naqvi, GM Hasan… - Current topics in …, 2020 - ingentaconnect.com
Microtubule-associated protein tau is involved in the tubulin binding leading to microtubule
stabilization in neuronal cells which is essential for stabilization of neuron cytoskeleton. The …

Virtual screening approach to identify high-affinity inhibitors of serum and glucocorticoid-regulated kinase 1 among bioactive natural products: Combined molecular …

T Mohammad, S Siddiqui, A Shamsi, MF Alajmi… - Molecules, 2020 - mdpi.com
Serum and glucocorticoid-regulated kinase 1 (SGK1) is a serine/threonine kinase that works
under acute transcriptional control by several stimuli, including serum and glucocorticoids. It …

[HTML][HTML] Ellagic acid controls cell proliferation and induces apoptosis in breast cancer cells via inhibition of cyclin-dependent kinase 6

M Yousuf, A Shamsi, P Khan, M Shahbaaz… - International journal of …, 2020 - mdpi.com
Cyclin-Dependent Kinase 6 (CDK6) plays an important role in cancer progression, and thus,
it is considered as an attractive drug target in anticancer therapeutics. This study presents an …

Identification and evaluation of bioactive natural products as potential inhibitors of human microtubule affinity-regulating kinase 4 (MARK4)

T Mohammad, FI Khan, KA Lobb, A Islam… - Journal of …, 2019 - Taylor & Francis
Microtubule affinity-regulating kinase 4 (MARK4) has recently been identified as a potential
drug target for several complex diseases including cancer, diabetes and neurodegenerative …

Investigation of molecular mechanism of recognition between citral and MARK4: A newer therapeutic approach to attenuate cancer cell progression

F Naz, FI Khan, T Mohammad, P Khan… - International journal of …, 2018 - Elsevier
Microtubule affinity regulating kinase 4 (MARK4) is a member of AMP-activated protein
kinase, found to be involved in apoptosis, inflammation and many other regulatory …

Elucidation of dietary polyphenolics as potential inhibitor of microtubule affinity regulating kinase 4: in silico and in vitro studies

P Khan, S Rahman, A Queen, S Manzoor, F Naz… - Scientific reports, 2017 - nature.com
Microtubule affinity regulating kinase 4 (MARK4) is a Ser/Thr kinase belonging to AMPK-like
family, has recently become an important drug target against cancer and neurodegenerative …

Identification of sphingosine kinase-1 inhibitors from bioactive natural products targeting cancer therapy

DS Jairajpuri, T Mohammad, K Adhikari, P Gupta… - ACS …, 2020 - ACS Publications
Sphingosine kinase 1 (SphK1) is an oncogenic lipid kinase that catalyzes the formation of
sphingosine-1-phosphate via phosphorylation of sphingosine and known to play a crucial …

Identification of potential inhibitors of calcium/calmodulin‐dependent protein kinase IV from bioactive phytoconstituents

P Gupta, S Khan, Z Fakhar, A Hussain… - Oxidative Medicine …, 2020 - Wiley Online Library
Calcium/calmodulin‐dependent protein kinase IV (CaMKIV) is an upstream regulator of
CaMKK‐CaMKIV signaling cascade that activates various transcription factors, thereby …

Evidence of vanillin binding to CAMKIV explains the anti-cancer mechanism in human hepatic carcinoma and neuroblastoma cells

H Naz, M Tarique, P Khan, S Luqman… - Molecular and cellular …, 2018 - Springer
Human calcium/calmodulin-dependent protein kinase IV (CAMKIV) is a member of Ser/Thr
kinase family, and is associated with different types of cancer and neurodegenerative …

High throughput screening, docking, and molecular dynamics studies to identify potential inhibitors of human calcium/calmodulin-dependent protein kinase IV

A Beg, FI Khan, KA Lobb, A Islam… - Journal of …, 2019 - Taylor & Francis
Calcium/calmodulin-dependent protein kinase IV (CAMKIV) is associated with many
diseases including cancer and neurodegenerative disorders and thus being considered as …