Beyond adiponectin and leptin: adipose tissue-derived mediators of inter-organ communication

JB Funcke, PE Scherer - Journal of lipid research, 2019 - ASBMB
The breakthrough discoveries of leptin and adiponectin more than two decades ago led to a
widespread recognition of adipose tissue as an endocrine organ. Many more adipose tissue …

Adipose organ development and remodeling

S Cinti - Comprehensive Physiology, 2018 - iris.univpm.it
During the last decades, research on adipose tissues has spread in parallel with the
extension of obesity. Several observations converged on the idea that adipose tissues are …

Development of phenothiazine hybrids with potential medicinal interest: a review

MC Posso, FC Domingues, S Ferreira, S Silvestre - Molecules, 2022 - mdpi.com
The molecular hybridization approach has been used to develop compounds with improved
efficacy by combining two or more pharmacophores of bioactive scaffolds. In this context …

Molecular pathways linking adipose innervation to insulin action in obesity and diabetes mellitus

A Guilherme, F Henriques, AH Bedard… - Nature Reviews …, 2019 - nature.com
Adipose tissue comprises adipocytes and many other cell types that engage in dynamic
crosstalk in a highly innervated and vascularized tissue matrix. Although adipose tissue has …

Immunotherapy for cardiovascular disease

E Lutgens, D Atzler, Y Döring, J Duchene… - European heart …, 2019 - academic.oup.com
The outcomes of the Canakinumab Anti-inflammatory Thrombosis Outcome Study
(CANTOS) trial have unequivocally proven that inflammation is a key driver of …

Toward an understanding of how immune cells control brown and beige adipobiology

F Villarroya, R Cereijo, J Villarroya, A Gavaldà-Navarro… - Cell metabolism, 2018 - cell.com
Immune cells were recently found to have an unexpected involvement in controlling the
thermogenic activity of brown and beige adipose tissue. Here, we review how macrophages …

[HTML][HTML] The therapeutic potential of second and third generation CB1R antagonists

R Cinar, MR Iyer, G Kunos - Pharmacology & therapeutics, 2020 - Elsevier
Endocannabinoids acting via CB 1 receptors (CB 1 R) play a critical role in regulating
energy homeostasis, which was the rationale for the pharmaceutical development of CB 1 R …

Neurobiology of cannabinoid receptor signaling

B Lutz - Dialogues in clinical neuroscience, 2020 - Taylor & Francis
The endocannabinoid system (ECS) is a highly versatile signaling system within the nervous
system. Despite its widespread localization, its functions within the context of distinct neural …

Reappraisal of Adipose Tissue Inflammation in Obesity

A Engin - Obesity and Lipotoxicity, 2024 - Springer
Chronic low-grade inflammation is a central component in the pathogenesis of obesity-
related expansion of adipose tissue and complications in other metabolic tissues. Five …

Monoacylglycerol lipase (MAGL) as a promising therapeutic target

A Gil-Ordóñez, M Martín-Fontecha… - Biochemical …, 2018 - Elsevier
Monoacylglycerol lipase (MAGL) has been characterized as the main enzyme responsible
for the inactivation of the most abundant brain endocannabinoid, 2-arachidonoylglycerol (2 …