Recent developments of gallic acid derivatives and their hybrids in medicinal chemistry: A review

NAAL Zahrani, RM El-Shishtawy, AM Asiri - European journal of medicinal …, 2020 - Elsevier
The leading cause of several degenerative diseases such as atherosclerosis, cancer, aging,
cardiovascular, and inflammatory diseases is oxidative stress, a consequence of …

Oral delivery of anticancer drugs: challenges and opportunities

K Thanki, RP Gangwal, AT Sangamwar… - Journal of controlled …, 2013 - Elsevier
The present report focuses on the various aspects of oral delivery of anticancer drugs. The
significance of oral delivery in cancer therapeutics has been highlighted which principally …

Synovial fibroblasts: key players in rheumatoid arthritis

LC Huber, O Distler, I Tarner, RE Gay, S Gay… - Rheumatology, 2006 - academic.oup.com
Rheumatoid arthritis (RA) is a chronic autoimmune-disease of unknown origin that primarily
affects the joints and ultimately leads to their destruction. The involvement of immune cells is …

Mechanism-based profiling of enzyme families

MJ Evans, BF Cravatt - Chemical reviews, 2006 - ACS Publications
Genome sequencing projects have ushered biological research into a new age where
scientists are confronted with the daunting undertaking of assigning functions to the full …

Metastasis review: from bench to bedside

AM Alizadeh, S Shiri, S Farsinejad - Tumor biology, 2014 - Springer
Cancer is the final result of uninhibited cell growth that involves an enormous group of
associated diseases. One major aspect of cancer is when cells attack adjacent components …

Advances in therapeutic targeting of cancer stem cells within the tumor microenvironment: an updated review

K Dzobo, DA Senthebane, C Ganz, NE Thomford… - Cells, 2020 - mdpi.com
Despite great strides being achieved in improving cancer patients' outcomes through better
therapies and combinatorial treatment, several hurdles still remain due to therapy …

Profiling the structural determinants of pyrrolidine derivative as gelatinases (MMP-2 and MMP-9) inhibitors using in silico approaches

K Tabti, I Ahmad, I Zafar, A Sbai, H Maghat… - … Biology and Chemistry, 2023 - Elsevier
Quantitative structure activity relationship (QSAR) studies on pyrrolidine derivatives have
been established using CoMFA, CoMSIA, and Hologram QSAR analysis to estimate the …

The role of endogenous and exogenous enzymes in chronic wounds: a focus on the implications of aberrant levels of both host and bacterial proteases in wound …

SM McCarty, CA Cochrane, PD Clegg… - Wound Repair and …, 2012 - Wiley Online Library
Cutaneous wound healing is orchestrated by a number of physiological pathways that
ultimately lead to reformation of skin integrity and the production of functional scar tissue …

The role of the tissue microenvironment in the regulation of cancer cell motility and invasion

J Brábek, CT Mierke, D Rösel, P Veselý… - Cell communication and …, 2010 - Springer
During malignant neoplastic progression the cells undergo genetic and epigenetic cancer-
specific alterations that finally lead to a loss of tissue homeostasis and restructuring of the …

Recent advances in MMP inhibitor design

JF Fisher, S Mobashery - Cancer and Metastasis Reviews, 2006 - Springer
The search for an MMP inhibitor with anticancer efficacy is a nearly three-decade endeavor.
This inhibitor is yet to be found. The reasons for this failure include shortcomings in the …