Potent acetylcholinesterase inhibitors: potential drugs for Alzheimer's disease
Alzheimer's disease (AD) is one of the cognitive or memory-related impairments occurring
with advancing age. Since its exact mechanism is not known, the full therapy has still not …
with advancing age. Since its exact mechanism is not known, the full therapy has still not …
LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes
Abstract Galanga (Alpinia officinarum Hance) is a pungent and aromatic rhizome, which is a
member of the ginger family (Zingiberaceae). The rhizomes of this plant have been used as …
member of the ginger family (Zingiberaceae). The rhizomes of this plant have been used as …
The first synthesis, carbonic anhydrase inhibition and anticholinergic activities of some bromophenol derivatives with S including natural products
Starting from vanillin, known four benzyl bromides with Br were synthesized. The first
synthesis of natural product 3, 4-dibromo-5-((methylsulfonyl) methyl) benzene-1, 2-diol (2) …
synthesis of natural product 3, 4-dibromo-5-((methylsulfonyl) methyl) benzene-1, 2-diol (2) …
Antioxidant and acetylcholinesterase inhibition properties of novel bromophenol derivatives
In this study, series of novel bromophenol derivatives were synthesized and investigated for
their antioxidant and AChE inhibition properties. Novel brominated diarylmethanones were …
their antioxidant and AChE inhibition properties. Novel brominated diarylmethanones were …
Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds–determination of their carbonic anhydrase, acetylcholinesterase …
Abstract Sulfur-containing pyrroles (1–3), tris (2-pyridyl) phosphine (selenide) sulfide (4–5)
and 4-benzyl-6-(thiophen-2-yl) pyrimidin-2-amine (6) were synthesized and characterized …
and 4-benzyl-6-(thiophen-2-yl) pyrimidin-2-amine (6) were synthesized and characterized …
Enzymatic assays for the assessment of toxic effects of halogenated organic contaminants in water and food. A review
AE Artabe, H Cunha-Silva, A Barranco - Food and Chemical Toxicology, 2020 - Elsevier
Halogenated organic compounds are a particular group of contaminants consisting of a
large number of substances, and of great concern due to their persistence in the …
large number of substances, and of great concern due to their persistence in the …
Synthesis and carbonic anhydrase isoenzymes I, II, IX, and XII inhibitory effects of dimethoxybromophenol derivatives incorporating cyclopropane moieties
M Boztas, Y Cetinkaya, M Topal, I Gulcin… - Journal of medicinal …, 2015 - ACS Publications
Cyclopropylcarboxylic acids and esters and cyclopropylmethanols incorporating
bromophenol moieties were investigated as inhibitors of the carbonic anhydrase enzyme …
bromophenol moieties were investigated as inhibitors of the carbonic anhydrase enzyme …
The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase …
Caffeic acid phenethyl ester (CAPE) is an active component of honeybee propolis extracts.
Carbonic anhydrases (CAs, EC 4.2. 1.1) are widespread and intensively studied …
Carbonic anhydrases (CAs, EC 4.2. 1.1) are widespread and intensively studied …
Novel antioxidant bromophenols with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions
In this study, a series of novel bromophenols were synthesized from benzoic acids and
methoxylated bromophenols. The synthesized compounds were evaluated by using different …
methoxylated bromophenols. The synthesized compounds were evaluated by using different …
Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds
In the present study a series of urea and sulfamide compounds incorporating the tetralin
scaffolds were synthesized and evaluated for their acetylcholinesterase (AChE), human …
scaffolds were synthesized and evaluated for their acetylcholinesterase (AChE), human …