[HTML][HTML] A review of biological targets and therapeutic approaches in the management of triple-negative breast cancer

H Kumar, NV Gupta, R Jain… - Journal of Advanced …, 2023 - Elsevier
Background Triple-negative breast cancer (TNBC) is a heterogeneous, aggressive
phenotype of breast cancer with associated chemoresistance. The development of chemo-or …

[HTML][HTML] HIF-1-independent mechanisms regulating metabolic adaptation in hypoxic cancer cells

SH Lee, M Golinska, JR Griffiths - Cells, 2021 - mdpi.com
In solid tumours, cancer cells exist within hypoxic microenvironments, and their metabolic
adaptation to this hypoxia is driven by HIF-1 transcription factor, which is overexpressed in a …

Exploration of 1, 2, 3-triazole linked benzenesulfonamide derivatives as isoform selective inhibitors of human carbonic anhydrase

C Kakakhan, C Türkeş, Ö Güleç, Y Demir… - Bioorganic & Medicinal …, 2023 - Elsevier
Abstract A novel series of 1, 2, 3-triazole benzenesulfonamide substituted 1, 3-
dioxoisoindolin-5-carboxylate (7a-l) inhibitors of human α-carbonic anhydrase (hCA) was …

A strategy of Fenton reaction cycloacceleration for high‐performance ferroptosis therapy initiated by tumor microenvironment remodeling

L Huang, J Feng, J Zhu, J Yang… - Advanced …, 2023 - Wiley Online Library
The emerging tumor ferroptosis therapy confronts impediments of the tumor
microenvironment (TME) with weak intrinsic acidity, inadequate endogenous H2O2, and a …

Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment

A Angeli, F Carta, A Nocentini, JY Winum… - Metabolites, 2020 - mdpi.com
The tumor microenvironment is crucial for the growth of cancer cells, triggering particular
biochemical and physiological changes, which frequently influence the outcome of …

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase

A Nocentini, A Angeli, F Carta, JY Winum… - Journal of Enzyme …, 2021 - Taylor & Francis
Inorganic anions inhibit the metalloenzyme carbonic anhydrase (CA, EC 4.2. 1.1) generally
by coordinating to the active site metal ion. Cyanate was reported as a non-coordinating CA …

Ratiometric fluorescent probes for pH map** in cellular organelles

S Munan, R Yadav, N Pareek, A Samanta - Analyst, 2023 - pubs.rsc.org
The intracellular pH (pHi) in organelles, including mitochondria, endoplasmic reticulum,
lysosomes, and nuclei, differs from the cytoplasmic pH, and thus maintaining the pH of these …

Drug delivery systems for localized cancer combination therapy

RN Woodring, EG Gurysh, EM Bachelder… - ACS applied bio …, 2023 - ACS Publications
With over 2 million cancer cases and over 600,000 cancer-associated deaths predicted in
the US for 2022, this life-debilitating disease continuously impacts the lives of people across …

Recent progress in magnetically actuated microrobots for targeted delivery of therapeutic agents

J Choi, J Hwang, J Kim, H Choi - Advanced Healthcare …, 2021 - Wiley Online Library
Therapeutic agents, such as drugs and cells, play an essential role in virtually every
treatment of injury, illness, or disease. However, the conventional practices of drug delivery …

Metabolic tricks of cancer cells

K Hönigova, J Navratil, B Peltanova… - … et Biophysica Acta (BBA …, 2022 - Elsevier
One of the characteristics of cancer cells important for tumorigenesis is their metabolic
plasticity. Indeed, in various stress conditions, cancer cells can reshape their metabolic …