[HTML][HTML] Recent Developments and Biological Activities of N-Substituted Carbazole Derivatives: A Review

M Bashir, A Bano, AS Ijaz, BA Chaudhary - Molecules, 2015 - mdpi.com
Carbazoles represent an important class of heterocycles. These have been reported to
exhibit diverse biological activities such as antimicrobial, antitumor, antiepileptic …

Phytocarbazoles: Alkaloids with great structural diversity and pronounced biological activities

H Greger - Phytochemistry reviews, 2017 - Springer
Carbazole alkaloids characterized by a heterocyclic aromatic basic skeleton are known from
different organisms but do not represent a biogenetically homogenous group. The majority …

Synthesis, antibacterial and antifungal activities of some carbazole derivatives

FF Zhang, LL Gan, CH Zhou - Bioorganic & medicinal chemistry letters, 2010 - Elsevier
A series of N-substituted carbazole derivatives were synthesized and evaluated for
antibacterial and antifungal activities against Staphylococcus aureus, methicillin-resistant …

Palladium-catalyzed triple successive C–H functionalization: direct synthesis of functionalized carbazoles from indoles

AK Verma, AK Danodia, RK Saunthwal, M Patel… - Organic …, 2015 - ACS Publications
A novel Pd (II)-catalyzed approach for the direct synthesis of differentially substituted
carbazoles from free (NH) indoles via regioselective triple successive oxidative Heck …

Potential Antimicrobial Isopropanol-Conjugated Carbazole Azoles as Dual Targeting Inhibitors of Enterococcus faecalis

Y Zhang, VKR Tangadanchu, Y Cheng… - ACS Medicinal …, 2018 - ACS Publications
A series of isopropanol-bridged carbazole azoles as potential antimicrobial agents were
designed and synthesized from commercial carbazoles. Bioassay revealed that 3, 6 …

A tandem approach to functionalized carbazoles from indoles via two successive regioselective oxidative Heck reactions followed by thermal electrocyclization

JK Laha, N Dayal - Organic Letters, 2015 - ACS Publications
A direct one-pot approach to the synthesis of carbazoles (mono-, di-, and trisubstituted) and
α-carbolines from readily available indoles or 7-azaindoles and alkenes is described. Based …

Design, Synthesis and In Vitro Characterization of Novel Antimicrobial Agents Based on 6-Chloro-9H-carbazol Derivatives and 1,3,4-Oxadiazole Scaffolds

AT Bordei Telehoiu, DC Nuță, MT Căproiu… - Molecules, 2020 - mdpi.com
In this paper, we aimed to exploit and combine in the same molecule the carbazole and the
1, 3, 4-oxadiazole pharmacophores, to obtain novel carprofen derivatives, by using two …

Natural carbazole alkaloid murrayafoline A displays potent anti-neuroinflammatory effect by directly targeting transcription factor Sp1 in LPS-induced microglial cells

CH Li, Y Zhou, PF Tu, KW Zeng, Y Jiang - Bioorganic Chemistry, 2022 - Elsevier
Neuroinflammation is a leading cause for neurological disorders. Carbazole alkaloids,
isolated from the medicinal plants of Murraya species (Rutaceae), have exhibited wide …

Conventional and microwave-assisted synthesis, antimicrobial and antioxidant activity evaluation with in silico studies of carbazole-thiazole-Schiff base hybrids

SS Marufa, MM Rahman, MM Rahman… - Journal of Molecular …, 2025 - Elsevier
Conventional and microwave irradiation (MWI) methods were applied to synthesize a series
of thirteen carbazole-thiazole-Schiff base hybrids (2a-2m). MWI assisted synthesis was a …

Iodine-catalyzed aromatization of tetrahydrocarbazoles and its utility in the synthesis of glycozoline and murrayafoline A: a combined experimental and computational …

V Humne, Y Dangat, K Vanka… - Organic & Biomolecular …, 2014 - pubs.rsc.org
A new protocol for the aromatization of tetrahydrocarbazoles has been achieved using a
catalytic amount of iodine, giving high yields. The role of iodine in the aromatization has …