Generating Robust and Informative Nonclinical In Vitro and In Vivo Bacterial Infection Model Efficacy Data To Support Translation to Humans

JB Bulitta, WW Hope, AE Eakin, T Guina… - Antimicrobial agents …, 2019 - Am Soc Microbiol
ABSTRACT In June 2017, the National Institute of Allergy and Infectious Diseases, part of
the National Institutes of Health, organized a workshop entitled “Pharmacokinetics …

Bacteriocin-antimicrobial synergy: a medical and food perspective

H Mathur, D Field, MC Rea, PD Cotter, C Hill… - Frontiers in …, 2017 - frontiersin.org
The continuing emergence of multi-drug resistant pathogens has sparked an interest in
seeking alternative therapeutic options. Antimicrobial combinatorial therapy is one such …

International consensus guidelines for the optimal use of the polymyxins: endorsed by the American college of clinical pharmacy (ACCP), European society of clinical …

BT Tsuji, JM Pogue, AP Zavascki… - … : The Journal of …, 2019 - Wiley Online Library
The polymyxin antibiotics colistin (polymyxin E) and polymyxin B became available in the
1950s and thus did not undergo contemporary drug development procedures. Their clinical …

Agents of last resort: polymyxin resistance

KS Kaye, JM Pogue, TB Tran, RL Nation… - Infectious Disease …, 2016 - id.theclinics.com
The polymyxins, colistin (also known as polymyxin E) and polymyxin B, have a unique and
interesting history. Originally introduced in the 1950s for the treatment of infections due to …

Limitations of antibiotic MIC-based PK-PD metrics: looking back to move forward

CB Landersdorfer, RL Nation - Frontiers in Pharmacology, 2021 - frontiersin.org
Within a few years after the first successful clinical use of penicillin, investigations were
conducted in animal infection models to explore a range of factors that were considered …

Polymyxin combination therapy for multidrug-resistant, extensively-drug resistant, and difficult-to-treat drug-resistant gram-negative infections: is it superior to …

A Ardebili, A Izanloo, M Rastegar - Expert Review of Anti-infective …, 2023 - Taylor & Francis
Introduction The increasing prevalence of infections with multidrug-resistant (MDR),
extensively-drug resistant (XDR) or difficult-to-treat drug resistant (DTR) Gram-negative …

Combination therapy for carbapenem-resistant Gram-negative bacteria

AP Zavascki, JB Bulitta… - Expert review of anti …, 2013 - Taylor & Francis
The emergence of resistant to carbapenems Gram-negative bacteria (CR GNB) has severely
challenged antimicrobial therapy. Many CR GNB isolates are only susceptible to …

Two mechanisms of killing of Pseudomonas aeruginosa by tobramycin assessed at multiple inocula via mechanism-based modeling

JB Bulitta, NS Ly, CB Landersdorfer… - Antimicrobial agents …, 2015 - Am Soc Microbiol
Bacterial resistance is among the most serious threats to human health globally, and many
bacterial isolates have emerged that are resistant to all antibiotics in monotherapy …

Mechanism of action of isopropoxy benzene guanidine against multidrug-resistant pathogens

J Li, X Zhang, N Han, P Wan, F Zhao, T Xu… - Microbiology …, 2023 - Am Soc Microbiol
The increasing emergence of antibiotic resistance is an urgent threat to global health care;
thus, there is a need for new therapeutics. Guanidine is the preferred functional group for …

Resveratrol enhances the antimicrobial effect of polymyxin B on Klebsiella pneumoniae and Escherichia coli isolates with polymyxin B resistance

L Liu, J Yu, X Shen, X Cao, Q Zhan, Y Guo, F Yu - BMC microbiology, 2020 - Springer
Abstract Background Multidrug resistant (MDR) Gram-negative bacterial infections are a
serious threat to human health due to the lack of effective treatments. In this study, we …